# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3664717 | BDBM107664 | IC50 | = | 4.3 | nM | ALA5245460 | 8.37 | nM | Mus musculus | ||
2. | ALA3664717 | BDBM107664 | INH | = | 95 | % | ALA4036219 | % | Macaca fascicularis | |||
3. | ALA3664717 | BDBM107664 | INH | = | 67 | % | ALA4036218 | % | Macaca fascicularis | |||
4. | ALA3664717 | BDBM107664 | INH | = | 90 | % | ALA4036217 | % | Macaca fascicularis | |||
5. | ALA3664717 | BDBM107664 | INH | = | 67 | % | ALA4036216 | % | Macaca fascicularis | |||
6. | ALA3664717 | BDBM107664 | Ratio IC50 | > | 1000 | ALA4036215 | ||||||
7. | ALA3664717 | BDBM107664 | Ratio IC50 | > | 1000 | ALA4036214 | ||||||
8. | ALA3664717 | BDBM107664 | Ratio IC50 | > | 1000 | ALA4036213 | ||||||
9. | ALA3664717 | BDBM107664 | Ratio IC50 | > | 1000 | ALA4036212 | ||||||
10. | ALA3664717 | BDBM107664 | CLH | = | 0.2 | ml/min.kg | ALA4036211 | mL.min-1.kg-1 | ||||
11. | ALA3664717 | BDBM107664 | PPB | = | 91.6 | % | ALA4036210 | % | Homo sapiens | |||
12. | ALA3664717 | BDBM107664 | logP | = | 2.6 | ALA4036209 | ||||||
13. | ALA3664717 | BDBM107664 | EC50 | > | 10 | uM | ALA4036208 | nM | Homo sapiens | |||
14. | ALA3664717 | BDBM107664 | IC50 | > | 10 | uM | ALA4036207 | nM | Homo sapiens | |||
15. | ALA3664717 | BDBM107664 | IC50 | > | 10 | uM | ALA4036206 | nM | Homo sapiens | |||
16. | ALA3664717 | BDBM107664 | IC50 | > | 10 | uM | ALA4036205 | nM | Homo sapiens | |||
17. | ALA3664717 | BDBM107664 | F | = | 54 | % | ALA4036204 | % | Macaca fascicularis | |||
18. | ALA3664717 | BDBM107664 | MRT | = | 8.7 | hr | ALA4036203 | hr | Macaca fascicularis | |||
19. | ALA3664717 | BDBM107664 | Vdss | = | 2.5 | L/Kg | ALA4036202 | L.kg-1 | Macaca fascicularis | |||
20. | ALA3664717 | BDBM107664 | CL | = | 7.5 | ml/min.kg | ALA4036201 | mL.min-1.kg-1 | Macaca fascicularis |