| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3675746 | BDBM123515 | IC50 | = | 0.114 | uM | ALA4178741 | 6.94 | nM | Homo sapiens | ||
| 2. | ALA3675746 | BDBM123515 | IC50 | = | 1 | uM | ALA4178742 | 6.00 | nM | Homo sapiens | ||
| 3. | ALA3675746 | BDBM123515 | Ratio IC50 | = | 9 | ALA4178743 | ||||||
| 4. | ALA3675746 | BDBM123515 | IC50 | = | 0.93 | uM | ALA4178744 | 6.03 | nM | Homo sapiens | ||
| 5. | ALA3675746 | BDBM123515 | IC50 | = | 55 | nM | ALA3705172 | 7.26 | 252433 | nM | Homo sapiens | |
| 6. | ALA3675746 | BDBM123515 | Activity | = | 4 | % | ALA4044446 | % | Mus musculus | |||
| 7. | ALA3675746 | BDBM123515 | Activity | = | 65 | % | ALA4044447 | % | Mus musculus | |||
| 8. | ALA3675746 | BDBM123515 | Activity | = | 94 | % | ALA4044448 | % | Mus musculus | |||
| 9. | ALA3675746 | BDBM123515 | Activity | = | 100 | % | ALA4044449 | % | Mus musculus | |||
| 10. | ALA3675746 | BDBM123515 | IC50 | = | 0.11 | uM | ALA4044420 | 6.96 | nM | Homo sapiens | ||
| 11. | ALA3675746 | BDBM123515 | IC50 | = | 1.29 | uM | ALA4044421 | 5.89 | nM | Mus musculus | ||
| 12. | ALA3675746 | BDBM123515 | IC50 | = | 0.8 | uM | ALA4044422 | 6.10 | nM | Rattus norvegicus | ||
| 13. | ALA3675746 | BDBM123515 | CL | = | 15 | ml/min.Kg | ALA4044425 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 14. | ALA3675746 | BDBM123515 | beta t1/2 | = | 5.6 | hr | ALA4044426 | hr | Rattus norvegicus | |||
| 15. | ALA3675746 | BDBM123515 | AUC/dose | = | 2196 | microg.min/mL | ALA4044427 | microg.min/mL | Rattus norvegicus | |||
| 16. | ALA3675746 | BDBM123515 | Cmax/dose | = | 193 | nM | ALA4044428 | nM | Rattus norvegicus | |||
| 17. | ALA3675746 | BDBM123515 | F | = | 86 | % | ALA4044429 | % | Rattus norvegicus | |||
| 18. | ALA3675746 | BDBM123515 | INH | 0 | ALA4044430 | Dose-dependent effect | % | Mus musculus | ||||
| 19. | ALA3675746 | BDBM123515 | INH | 0 | ALA4044431 | Dose-dependent effect | % | Rattus norvegicus | ||||
| 20. | ALA3675746 | BDBM123515 | INH | 0 | ALA4044432 | Active | % | Rattus norvegicus |
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