| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3681909 | BDBM141965 | Ki | = | 2.8 | nM | ALA3705528 | 8.55 | 277674 | nM | Homo sapiens | |
| 2. | ALA3681909 | BDBM141965 | F | = | 108 | % | ALA4355768 | % | ||||
| 3. | ALA3681909 | BDBM141965 | Vdss | = | 16.1 | L/Kg | ALA4355765 | L.kg-1 | ||||
| 4. | ALA3681909 | BDBM141965 | t1/2 | = | 4.03 | hr | ALA4355762 | hr | ||||
| 5. | ALA3681909 | BDBM141965 | CL | = | 45.8 | ml/min.kg | ALA4355760 | mL.min-1.kg-1 | ||||
| 6. | ALA3681909 | BDBM141965 | AUC/dose | = | 0.538 | uM.hr.kg/mg | ALA4355759 | uM.hr.kg/mg | ||||
| 7. | ALA3681909 | BDBM141965 | Ki | = | 4500 | nM | ALA4355756 | 5.35 | nM | Homo sapiens | ||
| 8. | ALA3681909 | BDBM141965 | EC50 | = | 152 | nM | ALA4355755 | 6.82 | nM | Rattus norvegicus | ||
| 9. | ALA3681909 | BDBM141965 | Ki | = | 2.8 | nM | ALA4355754 | 8.55 | nM | Homo sapiens | ||
| 10. | ALA3681909 | BDBM141965 | Papp | = | 0.8 | 10'-6 cm/s | ALA4355751 | 10'-6 cm/s |
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