# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3686863 | BDBM142234 | IC50 | = | 9.8 | nM | ALA3706135 | 8.01 | 278016 | nM | Homo sapiens | |
2. | ALA3686863 | BDBM142234 | Activity | 0 | ALA3795723 | Active | Rattus norvegicus | |||||
3. | ALA3686863 | BDBM142234 | solubility | = | 0.762 | mg/ml | ALA3796825 | ug.mL-1 | ||||
4. | ALA3686863 | BDBM142234 | AUC | = | 9670 | ng.hr/ml | ALA3796827 | ng.hr.mL-1 | Rattus norvegicus | |||
5. | ALA3686863 | BDBM142234 | Cmax | = | 3100 | ng/ml | ALA3796828 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
6. | ALA3686863 | BDBM142234 | t1/2 | = | 5.1 | hr | ALA3796829 | hr | Rattus norvegicus | |||
7. | ALA3686863 | BDBM142234 | F | = | 34 | % | ALA3796830 | % | Rattus norvegicus | |||
8. | ALA3686863 | BDBM142234 | Vdss | = | 0.34 | L/Kg | ALA3796831 | L.kg-1 | Rattus norvegicus | |||
9. | ALA3686863 | BDBM142234 | AUC | = | 6320 | ng.hr/ml | ALA3796832 | ng.hr.mL-1 | Canis lupus familiaris | |||
10. | ALA3686863 | BDBM142234 | Cmax | = | 1870 | ng/ml | ALA3796833 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Canis lupus familiaris | ||
11. | ALA3686863 | BDBM142234 | t1/2 | = | 5.1 | hr | ALA3796834 | hr | Canis lupus familiaris | |||
12. | ALA3686863 | BDBM142234 | CL | = | 10 | ml/min.kg | ALA3796835 | mL.min-1.kg-1 | Canis lupus familiaris | |||
13. | ALA3686863 | BDBM142234 | Vdss | = | 1.73 | L/Kg | ALA3796836 | L.kg-1 | Canis lupus familiaris | |||
14. | ALA3686863 | BDBM142234 | F | = | 75 | % | ALA3796837 | % | Canis lupus familiaris | |||
15. | ALA3686863 | BDBM142234 | IC50 | > | 10 | uM | ALA3795702 | nM | Homo sapiens | |||
16. | ALA3686863 | BDBM142234 | IC50 | > | 10 | uM | ALA3795703 | nM | Homo sapiens | |||
17. | ALA3686863 | BDBM142234 | IC50 | > | 10 | uM | ALA3795704 | nM | Homo sapiens | |||
18. | ALA3686863 | BDBM142234 | IC50 | > | 10 | uM | ALA3795705 | nM | Homo sapiens | |||
19. | ALA3686863 | BDBM142234 | IC50 | > | 10 | uM | ALA3795706 | nM | Homo sapiens | |||
20. | ALA3686863 | BDBM142234 | IC50 | > | 10 | uM | ALA3795707 | nM | Homo sapiens |