# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3746386 | 38; UR-MK299 | INH | 0 | ALA3750539 | Dose-dependent effect | % | Homo sapiens | ||||
2. | ALA3746386 | 38; UR-MK299 | INH | 0 | ALA3750348 | Dose-dependent effect | % | Homo sapiens | ||||
3. | ALA3746386 | 38; UR-MK299 | pIC50 | = | 9.49 | ALA3750540 | 9.49 | nM | Homo sapiens | |||
4. | ALA3746386 | 38; UR-MK299 | IC50 | = | 7.61 | nM | ALA3750539 | 8.12 | nM | Homo sapiens | ||
5. | ALA3746386 | 38; UR-MK299 | INH | <= | 90 | % | ALA3750539 | % | Homo sapiens | |||
6. | ALA3746386 | 38; UR-MK299 | INH | 0 | ALA3750539 | tde | % | Homo sapiens | ||||
7. | ALA3746386 | 38; UR-MK299 | Retention_time | = | 18.3 | min | ALA3750525 | min | ||||
8. | ALA3746386 | 38; UR-MK299 | Ki | > | 3000 | nM | ALA3750524 | nM | Homo sapiens | |||
9. | ALA3746386 | 38; UR-MK299 | Ki | = | 1000 | nM | ALA3750369 | 6.00 | nM | Homo sapiens | ||
10. | ALA3746386 | 38; UR-MK299 | Ki | > | 10000 | nM | ALA3750368 | nM | Homo sapiens | |||
11. | ALA3746386 | 38; UR-MK299 | Ki | > | 10000 | nM | ALA3750367 | nM | Homo sapiens | |||
12. | ALA3746386 | 38; UR-MK299 | Ki | > | 3000 | nM | ALA3750366 | nM | Homo sapiens | |||
13. | ALA3746386 | 38; UR-MK299 | Ki | = | 0.23 | nM | ALA3750365 | 9.64 | nM | Homo sapiens | ||
14. | ALA3746386 | 38; UR-MK299 | Ki | = | 0.077 | nM | ALA3750364 | 10.11 | nM | Homo sapiens | ||
15. | ALA3746386 | 38; UR-MK299 | Ki | = | 0.1 | nM | ALA3750362 | 10.00 | nM | Homo sapiens | ||
16. | ALA3746386 | 38; UR-MK299 | Ki | = | 0.31 | nM | ALA3750361 | 9.51 | nM | Homo sapiens | ||
17. | ALA3746386 | 38; UR-MK299 | pIC50 | = | 10 | ALA3750356 | 10.00 | nM | Homo sapiens | |||
18. | ALA3746386 | 38; UR-MK299 | pIC50 | = | 9.89 | ALA3750355 | 9.89 | nM | Homo sapiens | |||
19. | ALA3746386 | 38; UR-MK299 | pIC50 | = | 9.77 | ALA3750353 | 9.77 | nM | Homo sapiens | |||
20. | ALA3746386 | 38; UR-MK299 | pIC50 | = | 9.77 | ALA3750352 | 9.77 | nM | Homo sapiens |