# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3753495 | 6 | Activity | 0 | ALA3992938 | Active | Homo sapiens | |||||
2. | ALA3753495 | 6 | Activity | 0 | ALA3992937 | Active | Homo sapiens | |||||
3. | ALA3753495 | 6 | Activity | 0 | ALA3992936 | Dose-dependent effect | Homo sapiens | |||||
4. | ALA3753495 | 6 | Activity | 0 | ALA3992935 | Dose-dependent effect | Homo sapiens | |||||
5. | ALA3753495 | 6 | Activity | 0 | ALA3992934 | Active | Homo sapiens | |||||
6. | ALA3753495 | 6 | Activity | 0 | ALA3992933 | Dose-dependent effect | Homo sapiens | |||||
7. | ALA3753495 | 6 | Activity | 0 | ALA3992932 | Dose-dependent effect | Homo sapiens | |||||
8. | ALA3753495 | 6 | INH | = | 81.4 | % | ALA3992922 | % | Homo sapiens | |||
9. | ALA3753495 | 6 | INH | 0 | ALA3992923 | Active | % | Homo sapiens | ||||
10. | ALA3753495 | 6 | IC50 | = | 5.2 | uM | ALA3992924 | 5.28 | nM | Homo sapiens | ||
11. | ALA3753495 | 6 | IC50 | = | 9.6 | uM | ALA3992925 | 5.02 | nM | Homo sapiens | ||
12. | ALA3753495 | 6 | IC50 | = | 2.6 | uM | ALA3992926 | 5.58 | nM | Homo sapiens | ||
13. | ALA3753495 | 6 | IC50 | = | 2 | uM | ALA3992927 | 5.70 | nM | Homo sapiens | ||
14. | ALA3753495 | 6 | INH | 0 | ALA3992928 | Dose-dependent effect | % | Homo sapiens | ||||
15. | ALA3753495 | 6 | INH | 0 | ALA3992929 | Dose-dependent effect | % | Homo sapiens | ||||
16. | ALA3753495 | 6 | Activity | 0 | ALA3992930 | Dose-dependent effect | Homo sapiens | |||||
17. | ALA3753495 | 6 | Activity | 0 | ALA3992931 | Active | Homo sapiens | |||||
18. | ALA3753495 | 6 | INH | = | 52.9 | % | ALA3757756 | % | Rattus norvegicus | |||
19. | ALA3753495 | 6 | INH | = | 74.1 | % | ALA3757755 | % | Rattus norvegicus | |||
20. | ALA3753495 | 6 | INH | = | 77.3 | % | ALA3757754 | % | Rattus norvegicus |