# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3758877 | 20; GAT100 | EC50 | = | 2.09 | nM | ALA3760352 | 8.68 | nM | Homo sapiens | ||
2. | ALA3758877 | 20; GAT100 | Emax | = | 103 | % | ALA3760353 | % | Homo sapiens | |||
3. | ALA3758877 | 20; GAT100 | EC50 | = | 174 | nM | ALA3760354 | 6.76 | nM | Homo sapiens | ||
4. | ALA3758877 | 20; GAT100 | Emax | = | 111 | % | ALA3760355 | % | Homo sapiens | |||
5. | ALA3758877 | 20; GAT100 | INH | 0 | ALA3760356 | Dose-dependent effect | % | Mus musculus | ||||
6. | ALA3758877 | 20; GAT100 | Activity | 0 | ALA3760357 | Not Active | Mus musculus | |||||
7. | ALA3758877 | 20; GAT100 | Activity | 0 | ALA3760358 | Not Active | Mus musculus | |||||
8. | ALA3758877 | 20; GAT100 | Activity | 0 | ALA3760359 | Not Active | Homo sapiens | |||||
9. | ALA3758877 | 20; GAT100 | Activity | 0 | ALA3760360 | Not Active | Homo sapiens | |||||
10. | ALA3758877 | 20; GAT100 | EC50 | = | 19.6 | nM | ALA3760363 | 7.71 | nM | Homo sapiens | ||
11. | ALA3758877 | 20; GAT100 | Emax | = | 71.7 | % | ALA3760364 | % | Mus musculus | |||
12. | ALA3758877 | 20; GAT100 | Emax | = | 11.2 | % | ALA3760365 | % | Mus musculus | |||
13. | ALA3758877 | 20; GAT100 | EC50 | = | 27.3 | nM | ALA3760366 | 7.56 | nM | Mus musculus | ||
14. | ALA3758877 | 20; GAT100 | Emax | = | 87.8 | % | ALA3760367 | % | Mus musculus | |||
15. | ALA3758877 | 20; GAT100 | Emax | = | 116.5 | % | ALA3760368 | % | Homo sapiens | |||
16. | ALA3758877 | 20; GAT100 | Activity | 0 | ALA3760369 | tde | Homo sapiens | |||||
17. | ALA3758877 | 20; GAT100 | Ratio EC50 | = | 14 | ALA3760370 | Homo sapiens | |||||
18. | ALA3758877 | 20; GAT100 | FC | = | 2.25 | ALA3760371 | Homo sapiens | |||||
19. | ALA3758877 | 20; GAT100 | INH | 0 | ALA3760372 | Active | % | Homo sapiens |