| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3759901 | 13c | Ratio EC50 | > | 450 | ALA3762453 | ||||||
| 2. | ALA3759901 | 13c | EC50 | > | 10 | uM | ALA3762452 | nM | Homo sapiens | |||
| 3. | ALA3759901 | 13c | Ratio | = | 0.55 | ALA3762451 | ||||||
| 4. | ALA3759901 | 13c | Drug uptake | = | 120 | ng/g | ALA3762450 | ng/g | Rattus norvegicus | |||
| 5. | ALA3759901 | 13c | Cp | = | 217 | ng/ml | ALA3762449 | ng/ml | Rattus norvegicus | |||
| 6. | ALA3759901 | 13c | Vdss | = | 2.97 | L/Kg | ALA3762448 | L.kg-1 | Rattus norvegicus | |||
| 7. | ALA3759901 | 13c | CL | = | 65.5 | ml/min.kg | ALA3762447 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 8. | ALA3759901 | 13c | MRT | = | 45.4 | min | ALA3762446 | hr | Rattus norvegicus | |||
| 9. | ALA3759901 | 13c | t1/2 | = | 51.5 | min | ALA3762445 | hr | Rattus norvegicus | |||
| 10. | ALA3759901 | 13c | IC50 | > | 30 | uM | ALA3762444 | nM | Homo sapiens | |||
| 11. | ALA3759901 | 13c | IC50 | > | 30 | uM | ALA3762443 | nM | Homo sapiens | |||
| 12. | ALA3759901 | 13c | IC50 | > | 30 | uM | ALA3762442 | nM | Homo sapiens | |||
| 13. | ALA3759901 | 13c | IC50 | = | 6.3 | uM | ALA3762441 | 5.20 | nM | Homo sapiens | ||
| 14. | ALA3759901 | 13c | Fu | = | 0.272 | ALA3762440 | ||||||
| 15. | ALA3759901 | 13c | Fu | = | 0.001 | ALA3762439 | Rattus norvegicus | |||||
| 16. | ALA3759901 | 13c | Fu | < | 0.001 | ALA3762438 | ||||||
| 17. | ALA3759901 | 13c | CLH | = | 46.7 | ml/min.kg | ALA3762437 | mL.min-1.kg-1 | ||||
| 18. | ALA3759901 | 13c | CLH | = | 11.9 | ml/min.kg | ALA3762436 | mL.min-1.kg-1 | Homo sapiens | |||
| 19. | ALA3759901 | 13c | %max | = | 60 | % | ALA3762432 | % | Homo sapiens | |||
| 20. | ALA3759901 | 13c | pEC50 | = | 8.27 | ALA3762431 | 8.27 | nM | Homo sapiens |
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