# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3758435 | 13d | Ratio EC50 | > | 450 | ALA3762453 | ||||||
2. | ALA3758435 | 13d | EC50 | > | 10 | uM | ALA3762452 | nM | Homo sapiens | |||
3. | ALA3758435 | 13d | Ratio | = | 0.95 | ALA3762451 | ||||||
4. | ALA3758435 | 13d | Drug uptake | = | 147 | ng/g | ALA3762450 | ng/g | Rattus norvegicus | |||
5. | ALA3758435 | 13d | Cp | = | 0.97 | ng/ml | ALA3762449 | ng/ml | Rattus norvegicus | |||
6. | ALA3758435 | 13d | Vdss | = | 1.92 | L/Kg | ALA3762448 | L.kg-1 | Rattus norvegicus | |||
7. | ALA3758435 | 13d | CL | = | 62.6 | ml/min.kg | ALA3762447 | mL.min-1.kg-1 | Rattus norvegicus | |||
8. | ALA3758435 | 13d | MRT | = | 30.7 | min | ALA3762446 | hr | Rattus norvegicus | |||
9. | ALA3758435 | 13d | t1/2 | = | 38.9 | min | ALA3762445 | hr | Rattus norvegicus | |||
10. | ALA3758435 | 13d | IC50 | > | 30 | uM | ALA3762444 | nM | Homo sapiens | |||
11. | ALA3758435 | 13d | IC50 | > | 30 | uM | ALA3762443 | nM | Homo sapiens | |||
12. | ALA3758435 | 13d | IC50 | > | 30 | uM | ALA3762442 | nM | Homo sapiens | |||
13. | ALA3758435 | 13d | IC50 | > | 30 | uM | ALA3762441 | nM | Homo sapiens | |||
14. | ALA3758435 | 13d | Fu | = | 0.17 | ALA3762440 | ||||||
15. | ALA3758435 | 13d | Fu | = | 0.011 | ALA3762439 | Rattus norvegicus | |||||
16. | ALA3758435 | 13d | Fu | = | 0.03 | ALA3762438 | ||||||
17. | ALA3758435 | 13d | CLH | = | 52 | ml/min.kg | ALA3762437 | mL.min-1.kg-1 | ||||
18. | ALA3758435 | 13d | CLH | = | 6.72 | ml/min.kg | ALA3762436 | mL.min-1.kg-1 | Homo sapiens | |||
19. | ALA3758435 | 13d | %max | = | 81 | % | ALA3762432 | % | Homo sapiens | |||
20. | ALA3758435 | 13d | pEC50 | = | 7.71 | ALA3762431 | 7.71 | nM | Homo sapiens |