| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3764920 | (8S,9R)-57 | IC50 | = | 1.1 | nM | ALA3767923 | 8.96 | nM | Homo sapiens | ||
| 2. | ALA3764920 | (8S,9R)-57 | F | = | 14 | % | ALA3767720 | % | Rattus norvegicus | |||
| 3. | ALA3764920 | (8S,9R)-57 | AUC | = | 914 | ng.hr/ml | ALA3767721 | ng.hr.mL-1 | Rattus norvegicus | |||
| 4. | ALA3764920 | (8S,9R)-57 | Cmax | = | 126 | ng/ml | ALA3767722 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 5. | ALA3764920 | (8S,9R)-57 | Vdss | = | 4.5 | L/Kg | ALA3767723 | L.kg-1 | Rattus norvegicus | |||
| 6. | ALA3764920 | (8S,9R)-57 | CL | = | 26 | ml/min.kg | ALA3767724 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 7. | ALA3764920 | (8S,9R)-57 | beta t1/2 | = | 2.29 | hr | ALA3767725 | hr | Rattus norvegicus | |||
| 8. | ALA3764920 | (8S,9R)-57 | EC50 | = | 389 | nM | ALA3767929 | 6.41 | nM | |||
| 9. | ALA3764920 | (8S,9R)-57 | GI50 | = | 279 | nM | ALA3767927 | nM | Homo sapiens | |||
| 10. | ALA3764920 | (8S,9R)-57 | EC50 | = | 6.3 | nM | ALA3767926 | 8.20 | nM | Homo sapiens |
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