| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3764768 | 27n | Activity | 0 | ALA3768599 | Active | Homo sapiens | |||||
| 2. | ALA3764768 | 27n | INH | 0 | ALA3768597 | Dose-dependent effect | % | Homo sapiens | ||||
| 3. | ALA3764768 | 27n | INH | 0 | ALA3768596 | Dose-dependent effect | % | Homo sapiens | ||||
| 4. | ALA3764768 | 27n | IC50 | = | 1 | uM | ALA3768359 | 6.00 | nM | Homo sapiens | ||
| 5. | ALA3764768 | 27n | solubility | = | 18 | uM | ALA3768360 | nM | ||||
| 6. | ALA3764768 | 27n | EC50 | > | 13 | uM | ALA3768361 | nM | Homo sapiens | |||
| 7. | ALA3764768 | 27n | permeability | = | 432.5 | ucm/s | ALA3768362 | ucm/s | ||||
| 8. | ALA3764768 | 27n | t1/2 | = | 0.2 | hr | ALA3768363 | hr | ||||
| 9. | ALA3764768 | 27n | t1/2 | = | 1 | hr | ALA3768364 | hr | Rattus norvegicus | |||
| 10. | ALA3764768 | 27n | t1/2 | = | 1.1 | hr | ALA3768365 | hr | Homo sapiens | |||
| 11. | ALA3764768 | 27n | t1/2 | > | 4 | hr | ALA3768366 | hr | Canis lupus familiaris | |||
| 12. | ALA3764768 | 27n | CLH | = | 329.4 | ml/min.kg | ALA3768367 | mL.min-1.kg-1 | ||||
| 13. | ALA3764768 | 27n | CLH | = | 45.1 | ml/min.kg | ALA3768368 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 14. | ALA3764768 | 27n | CLH | = | 18.8 | ml/min.kg | ALA3768369 | mL.min-1.kg-1 | Homo sapiens | |||
| 15. | ALA3764768 | 27n | CLH | < | 7.9 | ml/min.kg | ALA3768370 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 16. | ALA3764768 | 27n | Stability | > | 24 | hr | ALA3768371 | hr | Mus musculus | |||
| 17. | ALA3764768 | 27n | Stability | > | 24 | hr | ALA3768372 | hr | Rattus norvegicus | |||
| 18. | ALA3764768 | 27n | Stability | > | 24 | hr | ALA3768374 | hr | Homo sapiens | |||
| 19. | ALA3764768 | 27n | PPB | 0 | ALA3768373 | Not Determined | % | |||||
| 20. | ALA3764768 | 27n | PPB | 0 | ALA3768375 | Not Determined | % |
The page will load shortly, Thanks for your patience!