# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3765335 | 22 | max activation | = | 91 | % | ALA3767597 | % | Macaca mulatta | |||
2. | ALA3765335 | 22 | max activation | = | 83 | % | ALA3767596 | % | Rattus norvegicus | |||
3. | ALA3765335 | 22 | max activation | = | 98 | % | ALA3767595 | % | Homo sapiens | |||
4. | ALA3765335 | 22 | max activation | = | 86 | % | ALA3766300 | % | Macaca fascicularis | |||
5. | ALA3765335 | 22 | EC50 | = | 39 | nM | ALA3766299 | 7.41 | nM | Canis lupus familiaris | ||
6. | ALA3765335 | 22 | Activity | 0 | ALA3768728 | Dose-dependent effect | Rattus norvegicus | |||||
7. | ALA3765335 | 22 | Activity | 0 | ALA3768727 | Dose-dependent effect | Rattus norvegicus | |||||
8. | ALA3765335 | 22 | EC50 | = | 2.1 | nM | ALA3768726 | 8.68 | nM | Homo sapiens | ||
9. | ALA3765335 | 22 | EC50 | = | 12 | nM | ALA3768725 | 7.92 | nM | Macaca mulatta | ||
10. | ALA3765335 | 22 | EC50 | = | 245 | nM | ALA3768724 | 6.61 | nM | Rattus norvegicus | ||
11. | ALA3765335 | 22 | max activation | = | 91 | % | ALA3768723 | % | Macaca mulatta | |||
12. | ALA3765335 | 22 | EC50 | = | 2.5 | nM | ALA3768722 | 8.60 | nM | Macaca mulatta | ||
13. | ALA3765335 | 22 | max activation | = | 85 | % | ALA3768721 | % | Rattus norvegicus | |||
14. | ALA3765335 | 22 | EC50 | = | 531 | nM | ALA3768720 | 6.28 | nM | Rattus norvegicus | ||
15. | ALA3765335 | 22 | IC50 | = | 2.3 | uM | ALA3768718 | 5.64 | nM | |||
16. | ALA3765335 | 22 | Ratio IC50/EC50 | > | 800 | ALA3768717 | ||||||
17. | ALA3765335 | 22 | Stability | = | 99 | % | ALA3768716 | % | Macaca mulatta | |||
18. | ALA3765335 | 22 | Stability | = | 77 | % | ALA3768715 | % | Canis lupus familiaris | |||
19. | ALA3765335 | 22 | Stability | = | 95 | % | ALA3768505 | % | Rattus norvegicus | |||
20. | ALA3765335 | 22 | Stability | = | 100 | % | ALA3768481 | % | Homo sapiens |