| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3763822 | (8S,9R)-36 | IC50 | = | 2.25 | nM | ALA3767923 | 8.65 | nM | Homo sapiens | ||
| 2. | ALA3763822 | (8S,9R)-36 | F | = | 91 | % | ALA3767720 | % | Rattus norvegicus | |||
| 3. | ALA3763822 | (8S,9R)-36 | AUC | = | 36500 | ng.hr/ml | ALA3767721 | ng.hr.mL-1 | Rattus norvegicus | |||
| 4. | ALA3763822 | (8S,9R)-36 | Cmax | = | 10530 | ng/ml | ALA3767722 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 5. | ALA3763822 | (8S,9R)-36 | Vdss | = | 0.5 | L/Kg | ALA3767723 | L.kg-1 | Rattus norvegicus | |||
| 6. | ALA3763822 | (8S,9R)-36 | CL | = | 4 | ml/min.kg | ALA3767724 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 7. | ALA3763822 | (8S,9R)-36 | beta t1/2 | = | 2.3 | hr | ALA3767725 | hr | Rattus norvegicus | |||
| 8. | ALA3763822 | (8S,9R)-36 | EC50 | = | 305 | nM | ALA3767929 | 6.52 | nM | |||
| 9. | ALA3763822 | (8S,9R)-36 | GI50 | = | 261 | nM | ALA3767927 | nM | Homo sapiens | |||
| 10. | ALA3763822 | (8S,9R)-36 | EC50 | = | 6.9 | nM | ALA3767926 | 8.16 | nM | Homo sapiens |
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