| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3764202 | (8S,9R)-42 | IC50 | = | 1.6 | nM | ALA3767923 | 8.80 | nM | Homo sapiens | ||
| 2. | ALA3764202 | (8S,9R)-42 | F | = | 68 | % | ALA3767720 | % | Rattus norvegicus | |||
| 3. | ALA3764202 | (8S,9R)-42 | AUC | = | 1810 | ng.hr/ml | ALA3767721 | ng.hr.mL-1 | Rattus norvegicus | |||
| 4. | ALA3764202 | (8S,9R)-42 | Cmax | = | 3988 | ng/ml | ALA3767722 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 5. | ALA3764202 | (8S,9R)-42 | Vdss | = | 0.73 | L/Kg | ALA3767723 | L.kg-1 | Rattus norvegicus | |||
| 6. | ALA3764202 | (8S,9R)-42 | CL | = | 6 | ml/min.kg | ALA3767724 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 7. | ALA3764202 | (8S,9R)-42 | beta t1/2 | = | 2.1 | hr | ALA3767725 | hr | Rattus norvegicus | |||
| 8. | ALA3764202 | (8S,9R)-42 | EC50 | = | 39 | nM | ALA3767929 | 7.41 | nM | |||
| 9. | ALA3764202 | (8S,9R)-42 | GI50 | = | 25 | nM | ALA3767927 | nM | Homo sapiens | |||
| 10. | ALA3764202 | (8S,9R)-42 | EC50 | = | 17.9 | nM | ALA3767926 | 7.75 | nM | Homo sapiens |
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