| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3764017 | 24 | F | = | 100 | % | ALA3768899 | % | Mus musculus | |||
| 2. | ALA3764017 | 24 | F | = | 88 | % | ALA3768898 | % | Mus musculus | |||
| 3. | ALA3764017 | 24 | Vdss | = | 7.42 | L/Kg | ALA3768897 | L.kg-1 | Mus musculus | |||
| 4. | ALA3764017 | 24 | CL | = | 168.7 | ml/min.kg | ALA3768896 | mL.min-1.kg-1 | Mus musculus | |||
| 5. | ALA3764017 | 24 | AUC | = | 5784 | nM.hr | ALA3768895 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 6. | ALA3764017 | 24 | AUC | = | 1516 | nM.hr | ALA3768888 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 7. | ALA3764017 | 24 | AUC | = | 173 | nM.hr | ALA3768894 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 8. | ALA3764017 | 24 | Tmax | = | 0.63 | hr | ALA3768893 | hr | Mus musculus | |||
| 9. | ALA3764017 | 24 | Tmax | = | 0.5 | hr | ALA3768892 | hr | Mus musculus | |||
| 10. | ALA3764017 | 24 | Cmax | = | 2863 | nM | ALA3768891 | nM | Mus musculus | |||
| 11. | ALA3764017 | 24 | Cmax | = | 941 | nM | ALA3768890 | nM | Mus musculus | |||
| 12. | ALA3764017 | 24 | Cmax | = | 274 | nM | ALA3768889 | nM | Mus musculus | |||
| 13. | ALA3764017 | 24 | t1/2 | = | 1.33 | hr | ALA3768887 | hr | Mus musculus | |||
| 14. | ALA3764017 | 24 | t1/2 | = | 0.99 | hr | ALA3768886 | hr | Mus musculus | |||
| 15. | ALA3764017 | 24 | t1/2 | = | 0.58 | hr | ALA3768885 | hr | Mus musculus | |||
| 16. | ALA3764017 | 24 | EC50 | = | 3 | uM | ALA3768884 | 5.52 | nM | Homo sapiens | ||
| 17. | ALA3764017 | 24 | Activity | = | 140 | % | ALA3768884 | % | Homo sapiens | |||
| 18. | ALA3764017 | 24 | IC50 | = | 9 | uM | ALA3768883 | 5.05 | nM | Homo sapiens | ||
| 19. | ALA3764017 | 24 | IC50 | = | 13 | uM | ALA3768882 | 4.89 | nM | Homo sapiens | ||
| 20. | ALA3764017 | 24 | IC50 | = | 3 | uM | ALA3768881 | 5.52 | nM | Homo sapiens |
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