# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3771118 | 4a; PF-06761281 | pIC50 | = | 6.9 | ALA3773098 | 6.90 | nM | Rattus norvegicus | |||
2. | ALA3771118 | 4a; PF-06761281 | pIC50 | = | 6.67 | ALA3773097 | 6.67 | nM | Mus musculus | |||
3. | ALA3771118 | 4a; PF-06761281 | pIC50 | = | 5 | ALA3773094 | 5.00 | nM | Homo sapiens | |||
4. | ALA3771118 | 4a; PF-06761281 | pIC50 | = | 5 | ALA3773093 | 5.00 | nM | Homo sapiens | |||
5. | ALA3771118 | 4a; PF-06761281 | pIC50 | = | 6.1 | ALA3773092 | 6.10 | nM | Homo sapiens | |||
6. | ALA3771118 | 4a; PF-06761281 | pIC50 | = | 6.3 | ALA3773091 | 6.30 | nM | Homo sapiens | |||
7. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773663 | Active | % | Mus musculus | ||||
8. | ALA3771118 | 4a; PF-06761281 | Therm_solubility | = | 24 | uM | ALA3773662 | nM | ||||
9. | ALA3771118 | 4a; PF-06761281 | Ratio IC50 | > | 25 | ALA3773661 | ||||||
10. | ALA3771118 | 4a; PF-06761281 | Ratio IC50 | > | 25 | ALA3773660 | ||||||
11. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773659 | Not Active | % | Homo sapiens | ||||
12. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773658 | Not Active | % | Homo sapiens | ||||
13. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773657 | Not Active | % | Homo sapiens | ||||
14. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773656 | Not Active | % | Homo sapiens | ||||
15. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773655 | Not Active | % | Homo sapiens | ||||
16. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773654 | Not Active | % | Homo sapiens | ||||
17. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773653 | Not Active | % | Homo sapiens | ||||
18. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773652 | Not Active | % | Homo sapiens | ||||
19. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773651 | Not Active | % | Homo sapiens | ||||
20. | ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773650 | Not Active | % | Homo sapiens |