# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3769849 | 7 | Ki | = | 80 | nM | ALA5123927 | 7.10 | nM | |||
2. | ALA3769849 | 7 | Ki | = | 180 | nM | ALA4735334 | 6.75 | nM | Homo sapiens | ||
3. | ALA3769849 | 7 | IC50 | = | 50.4 | nM | ALA3887471 | 7.30 | 340419 | nM | Homo sapiens | |
4. | ALA3769849 | 7 | IC50 | = | 41.8 | nM | ALA3887470 | 7.38 | 340357 | nM | Homo sapiens | |
5. | ALA3769849 | 7 | IC50 | = | 184.6 | nM | ALA3887469 | 6.73 | 340297 | nM | Homo sapiens | |
6. | ALA3769849 | 7 | IC50 | = | 260 | nM | ALA3887468 | 6.58 | 340235 | nM | Homo sapiens | |
7. | ALA3769849 | 7 | IC50 | > | 3 | uM | ALA3772963 | nM | Homo sapiens | |||
8. | ALA3769849 | 7 | solubility | 0 | ALA3772955 | soluble | ||||||
9. | ALA3769849 | 7 | F | = | 41 | % | ALA3772962 | % | Mus musculus | |||
10. | ALA3769849 | 7 | Vdss | = | 1.5 | L/Kg | ALA3772961 | L.kg-1 | Mus musculus | |||
11. | ALA3769849 | 7 | AUC | = | 950 | hr.ng/ml | ALA3772960 | ng.hr.mL-1 | Mus musculus | |||
12. | ALA3769849 | 7 | CL | = | 35 | ml/min.kg | ALA3772959 | mL.min-1.kg-1 | Mus musculus | |||
13. | ALA3769849 | 7 | EC50 | = | 10.5 | uM | ALA3772958 | 4.98 | nM | Homo sapiens | ||
14. | ALA3769849 | 7 | IC50 | = | 0.4 | uM | ALA3772956 | 6.40 | nM | Homo sapiens |