| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3770470 | 29 | AUC | = | 816 | ng.hr/ml | ALA3772645 | ng.hr.mL-1 | Rattus norvegicus | |||
| 2. | ALA3770470 | 29 | Tmax | = | 4 | hr | ALA3772644 | hr | Rattus norvegicus | |||
| 3. | ALA3770470 | 29 | Cmax | = | 102 | ng/ml | ALA3772643 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 4. | ALA3770470 | 29 | t1/2 | = | 3.1 | hr | ALA3772642 | hr | Rattus norvegicus | |||
| 5. | ALA3770470 | 29 | Ratio AUC | = | 2.9 | ALA3772637 | ||||||
| 6. | ALA3770470 | 29 | AUClast | = | 542 | ng.hr/ml | ALA3772636 | ng.hr.mL-1 | Mus musculus | |||
| 7. | ALA3770470 | 29 | AUClast | = | 286 | ng.hr/ml | ALA3772635 | ng.hr.mL-1 | Mus musculus | |||
| 8. | ALA3770470 | 29 | Cmax | = | 474 | ng/ml | ALA3772634 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 9. | ALA3770470 | 29 | Cmax | = | 130 | ng/ml | ALA3772633 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 10. | ALA3770470 | 29 | solubility | = | 2 | uM | ALA3772486 | nM | ||||
| 11. | ALA3770470 | 29 | logD | = | 1.92 | ALA3772485 | ||||||
| 12. | ALA3770470 | 29 | logD | > | 5 | ALA3772484 | ||||||
| 13. | ALA3770470 | 29 | Ki | = | 7.1 | uM | ALA3772483 | 5.15 | nM | Homo sapiens | ||
| 14. | ALA3770470 | 29 | Ki | = | 7.9 | uM | ALA3772472 | 5.10 | nM | Homo sapiens | ||
| 15. | ALA3770470 | 29 | Ki | > | 100 | uM | ALA3772482 | nM | Homo sapiens | |||
| 16. | ALA3770470 | 29 | Ki | = | 33 | uM | ALA3772481 | 4.48 | nM | Homo sapiens | ||
| 17. | ALA3770470 | 29 | Ki | = | 0.91 | uM | ALA3772480 | 6.04 | nM | Homo sapiens | ||
| 18. | ALA3770470 | 29 | Ki | = | 1.1 | uM | ALA3772479 | 5.96 | nM | |||
| 19. | ALA3770470 | 29 | Ki | = | 1.6 | uM | ALA3772478 | 5.80 | nM | Homo sapiens | ||
| 20. | ALA3770470 | 29 | Ki | = | 1.5 | uM | ALA3772477 | 5.82 | nM | Homo sapiens |
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