# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3774827 | 29 | beta t1/2 | = | 3.15 | hr | ALA3777106 | hr | Mus musculus | |||
2. | ALA3774827 | 29 | AUC | = | 1618 | nM.hr | ALA3777105 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
3. | ALA3774827 | 29 | Cmax | = | 535 | nM | ALA3777104 | nM | Mus musculus | |||
4. | ALA3774827 | 29 | Tmax | = | 0.83 | hr | ALA3777103 | hr | Mus musculus | |||
5. | ALA3774827 | 29 | IC50 | > | 10 | uM | ALA3777102 | nM | Homo sapiens | |||
6. | ALA3774827 | 29 | IC50 | > | 10 | uM | ALA3777101 | nM | Homo sapiens | |||
7. | ALA3774827 | 29 | IC50 | > | 15 | uM | ALA3777100 | nM | Homo sapiens | |||
8. | ALA3774827 | 29 | INH | 0 | ALA3777099 | Not Active | % | Homo sapiens | ||||
9. | ALA3774827 | 29 | INH | 0 | ALA3777098 | Not Active | % | Homo sapiens | ||||
10. | ALA3774827 | 29 | INH | 0 | ALA3777097 | Not Active | % | Homo sapiens | ||||
11. | ALA3774827 | 29 | Stability | = | 24.8 | % | ALA3777096 | % | ||||
12. | ALA3774827 | 29 | Stability | 0 | ALA3777092 | Not Determined | % | Canis lupus familiaris | ||||
13. | ALA3774827 | 29 | Stability | = | 80.7 | % | ALA3777093 | % | Homo sapiens | |||
14. | ALA3774827 | 29 | EC50 | = | 0.72 | uM | ALA3777094 | 6.14 | nM | Homo sapiens | ||
15. | ALA3774827 | 29 | IC50 | = | 0.06 | uM | ALA3777095 | 7.22 | nM | Homo sapiens |