# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3775940 | 36 | t1/2 | = | 66 | min | ALA3804162 | hr | Homo sapiens | |||
2. | ALA3775940 | 36 | t1/2 | = | 220 | min | ALA3804161 | hr | Homo sapiens | |||
3. | ALA3775940 | 36 | IC50 | > | 10 | uM | ALA3804160 | nM | Homo sapiens | |||
4. | ALA3775940 | 36 | IC50 | = | 0.044 | uM | ALA3804157 | 7.36 | nM | Homo sapiens | ||
5. | ALA3775940 | 36 | Selectivity ratio | = | 130 | ALA3804158 | ||||||
6. | ALA3775940 | 36 | IC50 | = | 2.1 | uM | ALA3804159 | 5.68 | nM | Homo sapiens | ||
7. | ALA3775940 | 36 | Ratio | = | 4.9 | ALA3776073 | ||||||
8. | ALA3775940 | 36 | Papp | = | 8.2 | ucm/s | ALA3776072 | ucm/s | ||||
9. | ALA3775940 | 36 | solubility | = | 100 | uM | ALA3776071 | nM | ||||
10. | ALA3775940 | 36 | CLH | = | 38.1 | uL/min | ALA3776070 | uL/min | Mus musculus | |||
11. | ALA3775940 | 36 | CLH | = | 28.2 | microL/min/mg | ALA3776069 | mL.min-1.g-1 | ||||
12. | ALA3775940 | 36 | CLH | = | 6.2 | microL/min/mg | ALA3776068 | mL.min-1.g-1 | Homo sapiens | |||
13. | ALA3775940 | 36 | t1/2 | = | 2 | hr | ALA3776067 | hr | Mus musculus | |||
14. | ALA3775940 | 36 | F | = | 35 | % | ALA3776066 | % | Mus musculus | |||
15. | ALA3775940 | 36 | IC50 | > | 10000 | nM | ALA3776065 | nM | ||||
16. | ALA3775940 | 36 | CLH | = | 20.9 | uL/min | ALA3776064 | uL/min | Mus musculus | |||
17. | ALA3775940 | 36 | Ratio IC50 | >= | 5 | ALA3776063 | ||||||
18. | ALA3775940 | 36 | IC50 | > | 10000 | nM | ALA3778241 | nM | Homo sapiens | |||
19. | ALA3775940 | 36 | IC50 | = | 2100 | nM | ALA3778240 | 5.68 | nM | Homo sapiens | ||
20. | ALA3775940 | 36 | Ratio IC50 | = | 130 | ALA3778239 |