# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3781751 | 22; ORY1001/RG-6016 | Ki | = | 50 | nM | ALA3887191 | 7.30 | 321815 | nM | Homo sapiens | |
2. | ALA3781751 | 22; ORY1001/RG-6016 | Ki | > | 40000 | nM | ALA3887028 | 321804 | nM | Homo sapiens | ||
3. | ALA3781751 | 22; ORY1001/RG-6016 | Ki | > | 40000 | nM | ALA3887027 | 3916 | nM | Homo sapiens | ||
4. | ALA3781751 | 22; ORY1001/RG-6016 | Selectivity index | = | 1 | ALA4513085 | Selectivity Index = Cc50/Ic50 | |||||
5. | ALA3781751 | 22; ORY1001/RG-6016 | CC50 | > | 33 | uM | ALA4513084 | nM | Chlorocebus sabaeus | |||
6. | ALA3781751 | 22; ORY1001/RG-6016 | IC50 | > | 33 | uM | ALA4513083 | nM | Severe acute respiratory syndrome coronavirus 2 | |||
7. | ALA3781751 | 22; ORY1001/RG-6016 | inhibition | = | 0.3 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
8. | ALA3781751 | 22; ORY1001/RG-6016 | Inhibition | = | 5.96 | % | ALA4495582 | % | Severe acute respiratory syndrome coronavirus 2 | |||
9. | ALA3781751 | 22; ORY1001/RG-6016 | CC50 | > | 33 | uM | ALA4513084 | nM | Chlorocebus sabaeus | |||
10. | ALA3781751 | 22; ORY1001/RG-6016 | IC50 | > | 33 | uM | ALA4513083 | nM | Severe acute respiratory syndrome coronavirus 2 | |||
11. | ALA3781751 | 22; ORY1001/RG-6016 | Selectivity index | = | 1 | ALA4513085 | Selectivity Index = Cc50/Ic50 | |||||
12. | ALA3781751 | 22; ORY1001/RG-6016 | inhibition | = | 0.3 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
13. | ALA3781751 | 22; ORY1001/RG-6016 | INH | = | 70 | % | ALA4008813 | % | Homo sapiens | |||
14. | ALA3781751 | 22; ORY1001/RG-6016 | Activity | 0 | ALA4008811 | Not Active | Homo sapiens | |||||
15. | ALA3781751 | 22; ORY1001/RG-6016 | Activity | 0 | ALA4008809 | Not Active | Homo sapiens | |||||
16. | ALA3781751 | 22; ORY1001/RG-6016 | FC | = | 54.8 | ALA4008802 | Homo sapiens | |||||
17. | ALA3781751 | 22; ORY1001/RG-6016 | FC | = | 11.1 | ALA4008800 | Homo sapiens | |||||
18. | ALA3781751 | 22; ORY1001/RG-6016 | FC | = | 5 | ALA4008798 | Homo sapiens | |||||
19. | ALA3781751 | 22; ORY1001/RG-6016 | IC50 | = | 12.9 | uM | ALA4008796 | 4.89 | nM | Homo sapiens | ||
20. | ALA3781751 | 22; ORY1001/RG-6016 | IC50 | > | 100 | uM | ALA4008795 | nM | Homo sapiens |