| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3781751 | 22; ORY1001/RG-6016 | Ki | = | 18 | nM | ALA5232456 | 7.75 | nM | Homo sapiens | ||
| 2. | ALA3781751 | 22; ORY1001/RG-6016 | Ratio IC50 | > | 1000 | ALA5159751 | ||||||
| 3. | ALA3781751 | 22; ORY1001/RG-6016 | Ratio IC50 | > | 1000 | ALA5159750 | ||||||
| 4. | ALA3781751 | 22; ORY1001/RG-6016 | Ratio IC50 | > | 1000 | ALA5159749 | ||||||
| 5. | ALA3781751 | 22; ORY1001/RG-6016 | IC50 | = | 0.018 | uM | ALA5159743 | 7.75 | nM | Homo sapiens | ||
| 6. | ALA3781751 | 22; ORY1001/RG-6016 | Activity | 0 | ALA4220810 | Toxic | Mus musculus | |||||
| 7. | ALA3781751 | 22; ORY1001/RG-6016 | Activity | 0 | ALA4220809 | Active | Mus musculus | |||||
| 8. | ALA3781751 | 22; ORY1001/RG-6016 | Activity | 0 | ALA4220808 | Active | Homo sapiens | |||||
| 9. | ALA3781751 | 22; ORY1001/RG-6016 | Activity | 0 | ALA4220807 | Active | Homo sapiens | |||||
| 10. | ALA3781751 | 22; ORY1001/RG-6016 | CC50 | > | 33 | uM | ALA4513084 | nM | Chlorocebus sabaeus | |||
| 11. | ALA3781751 | 22; ORY1001/RG-6016 | IC50 | > | 33 | uM | ALA4513083 | nM | Severe acute respiratory syndrome coronavirus 2 | |||
| 12. | ALA3781751 | 22; ORY1001/RG-6016 | Selectivity index | = | 1 | ALA4513085 | Selectivity Index = Cc50/Ic50 | |||||
| 13. | ALA3781751 | 22; ORY1001/RG-6016 | inhibition | = | 0.3 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
| 14. | ALA3781751 | 22; ORY1001/RG-6016 | INH | = | 70 | % | ALA4008813 | % | Homo sapiens | |||
| 15. | ALA3781751 | 22; ORY1001/RG-6016 | Activity | 0 | ALA4008811 | Not Active | Homo sapiens | |||||
| 16. | ALA3781751 | 22; ORY1001/RG-6016 | Activity | 0 | ALA4008809 | Not Active | Homo sapiens | |||||
| 17. | ALA3781751 | 22; ORY1001/RG-6016 | FC | = | 54.8 | ALA4008802 | Homo sapiens | |||||
| 18. | ALA3781751 | 22; ORY1001/RG-6016 | FC | = | 11.1 | ALA4008800 | Homo sapiens | |||||
| 19. | ALA3781751 | 22; ORY1001/RG-6016 | FC | = | 5 | ALA4008798 | Homo sapiens | |||||
| 20. | ALA3781751 | 22; ORY1001/RG-6016 | IC50 | = | 12.9 | uM | ALA4008796 | 4.89 | nM | Homo sapiens |
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