# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3786973 | 13 | Fu | = | 0.31 | ALA3789156 | ||||||
2. | ALA3786973 | 13 | Ki | > | 1000 | nM | ALA3789160 | nM | Homo sapiens | |||
3. | ALA3786973 | 13 | Fu | = | 34 | ng/ml | ALA3789159 | ng/ml | ||||
4. | ALA3786973 | 13 | Cmax | = | 1100 | ng/ml | ALA3789158 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
5. | ALA3786973 | 13 | LED | = | 20 | mg kg-1 | ALA3789157 | mg kg-1 | Rattus norvegicus | |||
6. | ALA3786973 | 13 | Ratio | = | 0.1 | ALA3789155 | ||||||
7. | ALA3786973 | 13 | F | = | 18 | % | ALA3789154 | % | Rattus norvegicus | |||
8. | ALA3786973 | 13 | CL | = | 26 | ml/min.kg | ALA3789153 | mL.min-1.kg-1 | Rattus norvegicus | |||
9. | ALA3786973 | 13 | Tmax | = | 0.5 | hr | ALA3789152 | hr | Rattus norvegicus | |||
10. | ALA3786973 | 13 | Tmax | = | 0.5 | hr | ALA3789151 | hr | Rattus norvegicus | |||
11. | ALA3786973 | 13 | logD | = | 1 | ALA3789150 | ||||||
12. | ALA3786973 | 13 | Ki | > | 1000 | nM | ALA3789149 | nM | ||||
13. | ALA3786973 | 13 | Ki | > | 1000 | nM | ALA3789148 | nM | ||||
14. | ALA3786973 | 13 | Ki | > | 1000 | nM | ALA3789147 | nM | Homo sapiens | |||
15. | ALA3786973 | 13 | Ki | > | 1000 | nM | ALA3789146 | nM | Homo sapiens | |||
16. | ALA3786973 | 13 | pIC50 | < | 5 | ALA3789145 | nM | Homo sapiens | ||||
17. | ALA3786973 | 13 | CLH | = | 8 | uL/min | ALA3789144 | uL/min | Homo sapiens | |||
18. | ALA3786973 | 13 | CLH | = | 33 | uL/min | ALA3789143 | uL/min | ||||
19. | ALA3786973 | 13 | Ki | = | 10 | nM | ALA3789139 | 8.00 | nM | Homo sapiens | ||
20. | ALA3786973 | 13 | pA2 | = | 8.4 | ALA3789140 | 8.40 | nM | Homo sapiens |