# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3787515 | 6a | Activity | 0 | ALA3792106 | Not Active | Rattus norvegicus | |||||
2. | ALA3787515 | 6a | Activity | 0 | ALA3792105 | Active | Rattus norvegicus | |||||
3. | ALA3787515 | 6a | Activity | = | 101 | mg | ALA3790123 | mg | Rattus norvegicus | |||
4. | ALA3787515 | 6a | F | = | 10 | % | ALA3792103 | % | Rattus norvegicus | |||
5. | ALA3787515 | 6a | AUC | = | 99 | ng/mL.hr | ALA3792102 | ng.hr.mL-1 | Rattus norvegicus | |||
6. | ALA3787515 | 6a | Tmax | = | 1.2 | hr | ALA3792101 | hr | Rattus norvegicus | |||
7. | ALA3787515 | 6a | Cmax | = | 25.2 | ng/ml | ALA3792100 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
8. | ALA3787515 | 6a | t1/2 | = | 2.5 | hr | ALA3790398 | hr | Rattus norvegicus | |||
9. | ALA3787515 | 6a | CL | = | 18.8 | ml/min.kg | ALA3790129 | mL.min-1.kg-1 | Rattus norvegicus | |||
10. | ALA3787515 | 6a | AUC | = | 996 | ng/mL.hr | ALA3790397 | ng.hr.mL-1 | Rattus norvegicus | |||
11. | ALA3787515 | 6a | Vdss | = | 2.7 | L/Kg | ALA3790128 | L.kg-1 | Rattus norvegicus | |||
12. | ALA3787515 | 6a | t1/2 | = | 3.2 | hr | ALA3790127 | hr | Rattus norvegicus | |||
13. | ALA3787515 | 6a | Ratio EC50 | = | 34 | ALA3790126 | ||||||
14. | ALA3787515 | 6a | EC50 | = | 42 | nM | ALA3790124 | 7.38 | nM | Homo sapiens | ||
15. | ALA3787515 | 6a | EC50 | = | 1412 | nM | ALA3790125 | 5.85 | nM | Homo sapiens |