# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3794064 | 3; BMS-520 | Ratio | = | 3 | ALA4681128 | ||||||
2. | ALA3794064 | 3; BMS-520 | Cp | = | 700 | nM | ALA4681127 | nM | ||||
3. | ALA3794064 | 3; BMS-520 | Activity | = | 91 | % | ALA4681126 | % | Rattus norvegicus | |||
4. | ALA3794064 | 3; BMS-520 | Cp | = | 2100 | nM | ALA4681125 | nM | ||||
5. | ALA3794064 | 3; BMS-520 | Activity | = | 78 | % | ALA4681124 | % | Rattus norvegicus | |||
6. | ALA3794064 | 3; BMS-520 | Ratio EC50 | = | 3400 | ALA4681123 | ||||||
7. | ALA3794064 | 3; BMS-520 | EC50 | = | 1600 | nM | ALA4681122 | 5.80 | nM | Homo sapiens | ||
8. | ALA3794064 | 3; BMS-520 | EC50 | = | 0.47 | nM | ALA4681121 | 9.33 | nM | Homo sapiens | ||
9. | ALA3794064 | 3; BMS-520 | ED50 | = | 0.02 | mg kg-1 | ALA3801548 | mg.kg-1 | Mus musculus | |||
10. | ALA3794064 | 3; BMS-520 | INH | 0 | ALA3801547 | Dose-dependent effect | % | Mus musculus | ||||
11. | ALA3794064 | 3; BMS-520 | INH | 0 | ALA3801546 | Dose-dependent effect | % | Mus musculus | ||||
12. | ALA3794064 | 3; BMS-520 | Activity | 0 | ALA3801544 | Dose-dependent effect | Mus musculus | |||||
13. | ALA3794064 | 3; BMS-520 | Activity | 0 | ALA3801543 | Dose-dependent effect | Mus musculus | |||||
14. | ALA3794064 | 3; BMS-520 | INH | 0 | ALA3801542 | Dose-dependent effect | % | Rattus norvegicus | ||||
15. | ALA3794064 | 3; BMS-520 | INH | 0 | ALA3801541 | Dose-dependent effect | % | Rattus norvegicus | ||||
16. | ALA3794064 | 3; BMS-520 | ED50 | = | 0.05 | mg kg-1 | ALA3801341 | mg.kg-1 | Rattus norvegicus | |||
17. | ALA3794064 | 3; BMS-520 | Activity | 0 | ALA3801342 | Active | Rattus norvegicus | |||||
18. | ALA3794064 | 3; BMS-520 | Activity | > | 50 | % | ALA3801540 | % | Rattus norvegicus | |||
19. | ALA3794064 | 3; BMS-520 | Activity | 0 | ALA3801343 | Not Active | Rattus norvegicus | |||||
20. | ALA3794064 | 3; BMS-520 | Ratio | = | 9 | ALA3801340 | Canis lupus familiaris |