# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3800086 | 20a | CL | = | 14600 | ml/min.kg | ALA3803491 | mL.min-1.kg-1 | Rattus norvegicus | |||
2. | ALA3800086 | 20a | CL/F | = | 275 | ml/min.kg | ALA3803477 | mL.min-1.kg-1 | Rattus norvegicus | |||
3. | ALA3800086 | 20a | Cp | < | 4 | ng/ml | ALA3803488 | ng/ml | Rattus norvegicus | |||
4. | ALA3800086 | 20a | Cp | = | 31 | ng/ml | ALA3803487 | ng/ml | Rattus norvegicus | |||
5. | ALA3800086 | 20a | Cp | = | 106 | ng/ml | ALA3803486 | ng/ml | Rattus norvegicus | |||
6. | ALA3800086 | 20a | Activity | = | 5 | % | ALA3803474 | % | Rattus norvegicus | |||
7. | ALA3800086 | 20a | Activity | = | -56 | % | ALA3803475 | % | Rattus norvegicus | |||
8. | ALA3800086 | 20a | Activity | = | -64 | % | ALA3803476 | % | Rattus norvegicus | |||
9. | ALA3800086 | 20a | CL free | = | 8100 | microL/min/mg | ALA3803483 | mL.min-1.g-1 | Rattus norvegicus | |||
10. | ALA3800086 | 20a | Fu | = | 0.012 | ALA3803482 | Rattus norvegicus | |||||
11. | ALA3800086 | 20a | Fu | = | 0.15 | ALA3803481 | Rattus norvegicus | |||||
12. | ALA3800086 | 20a | logD | = | 3.2 | ALA3803480 | ||||||
13. | ALA3800086 | 20a | CLH(app) | = | 1215 | microL/min/mg | ALA3803479 | mL.min-1.g-1 | Rattus norvegicus | |||
14. | ALA3800086 | 20a | Ratio EC50 | = | 733 | ALA3803478 | ||||||
15. | ALA3800086 | 20a | EC50 | = | 660 | nM | ALA3803472 | 6.18 | nM | Homo sapiens | ||
16. | ALA3800086 | 20a | EC50 | = | 0.9 | nM | ALA3803473 | 9.05 | nM | Homo sapiens |