Activities

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Activities

Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	ALA3799553	9u; TAK-259	Ratio Ki	=	200		ALA3801622
2.	ALA3799553	9u; TAK-259	INH		0		ALA3801635		Dose-dependent effect	%	Rattus norvegicus
3.	ALA3799553	9u; TAK-259	INH		0		ALA3801634		Dose-dependent effect	%	Rattus norvegicus
4.	ALA3799553	9u; TAK-259	MED	=	10	ug/kg	ALA3801636			ug/kg	Rattus norvegicus
5.	ALA3799553	9u; TAK-259	ID50	=	1.3	ug/kg	ALA3801635			mg.kg-1	Rattus norvegicus
6.	ALA3799553	9u; TAK-259	IC30	=	12	nM	ALA3801634			nM	Rattus norvegicus
7.	ALA3799553	9u; TAK-259	F	=	84.5	%	ALA3801633			%	Rattus norvegicus
8.	ALA3799553	9u; TAK-259	Ratio Ki	=	800		ALA3801623
9.	ALA3799553	9u; TAK-259	INH	=	16	%	ALA3801624			%	Homo sapiens
10.	ALA3799553	9u; TAK-259	Vdss	=	4432	ml/kg	ALA3801628			L.kg-1	Rattus norvegicus
11.	ALA3799553	9u; TAK-259	CL	=	2395	ml/hr/kg	ALA3801629			mL.min-1.kg-1	Rattus norvegicus
12.	ALA3799553	9u; TAK-259	Cmax	=	60.2	ng/ml	ALA3801630		standard_value was converted from ug.mL-1 to nM using the parent compound MW \| standard_value was converted from ug.mL-1 to nM using the parent compound MW \| standard_value was converted from ug.mL-1 to nM using the parent compound MW \| standard_value was converted from ug.mL-1 to nM using the parent compound MW \| standard_value was converted from ug.mL-1 to nM using the parent compound MW \| standard_value was converted from ug.mL-1 to nM using the parent compound MW	nM	Rattus norvegicus
13.	ALA3799553	9u; TAK-259	AUC	=	358	ng.hr/ml	ALA3801631			ng.hr.mL-1	Rattus norvegicus
14.	ALA3799553	9u; TAK-259	MRT	=	4.53	hr	ALA3801632			hr	Rattus norvegicus
15.	ALA3799553	9u; TAK-259	Ki	=	1.1	nM	ALA3801620	8.96		nM	Homo sapiens