# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3800282 | 5c | INH | < | 10 | % | ALA3802093 | % | Homo sapiens | |||
2. | ALA3800282 | 5c | INH | < | 10 | % | ALA3802092 | % | Homo sapiens | |||
3. | ALA3800282 | 5c | INH | < | 10 | % | ALA3802091 | % | Homo sapiens | |||
4. | ALA3800282 | 5c | Ratio | = | 0.6 | ALA3802089 | ||||||
5. | ALA3800282 | 5c | PPB | = | 99.3 | % | ALA3802088 | % | Rattus norvegicus | |||
6. | ALA3800282 | 5c | Drug uptake | = | 0.01 | uM | ALA3802086 | uM | Rattus norvegicus | |||
7. | ALA3800282 | 5c | Cp | = | 0.97 | uM | ALA3802085 | uM | Rattus norvegicus | |||
8. | ALA3800282 | 5c | AUC | = | 0.01 | uM.hr | ALA3802084 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
9. | ALA3800282 | 5c | Cmax | = | 0.12 | uM | ALA3802083 | nM | Rattus norvegicus | |||
10. | ALA3800282 | 5c | F | = | 0.2 | % | ALA3802082 | % | Rattus norvegicus | |||
11. | ALA3800282 | 5c | t1/2 | = | 1.2 | hr | ALA3802081 | hr | Rattus norvegicus | |||
12. | ALA3800282 | 5c | CL | = | 95.5 | ml/min.kg | ALA3804655 | mL.min-1.kg-1 | Rattus norvegicus | |||
13. | ALA3800282 | 5c | Ki | = | 94 | nM | ALA3804654 | 7.03 | nM | Homo sapiens | ||
14. | ALA3800282 | 5c | Ki | = | 389 | nM | ALA3804653 | 6.41 | nM | Homo sapiens |