# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3799347 | 3b | INH | = | 45 | % | ALA3802093 | % | Homo sapiens | |||
2. | ALA3799347 | 3b | INH | = | 55 | % | ALA3802092 | % | Homo sapiens | |||
3. | ALA3799347 | 3b | INH | = | 40 | % | ALA3802091 | % | Homo sapiens | |||
4. | ALA3799347 | 3b | CL | = | 6500 | ml/min.kg | ALA3802087 | mL.min-1.kg-1 | Rattus norvegicus | |||
5. | ALA3799347 | 3b | Drug uptake | = | 0.05 | uM | ALA3802086 | uM | Rattus norvegicus | |||
6. | ALA3799347 | 3b | Cp | = | 2.33 | uM | ALA3802085 | uM | Rattus norvegicus | |||
7. | ALA3799347 | 3b | AUC | = | 3.8 | uM.hr | ALA3802084 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
8. | ALA3799347 | 3b | Cmax | = | 1.6 | uM | ALA3802083 | nM | Rattus norvegicus | |||
9. | ALA3799347 | 3b | F | = | 33 | % | ALA3802082 | % | Rattus norvegicus | |||
10. | ALA3799347 | 3b | t1/2 | = | 6.5 | hr | ALA3802081 | hr | Rattus norvegicus | |||
11. | ALA3799347 | 3b | CL | = | 56 | ml/min.kg | ALA3804655 | mL.min-1.kg-1 | Rattus norvegicus | |||
12. | ALA3799347 | 3b | Ki | = | 189 | nM | ALA3804654 | 6.72 | nM | Homo sapiens | ||
13. | ALA3799347 | 3b | Ki | = | 312 | nM | ALA3804653 | 6.51 | nM | Homo sapiens |