| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3800053 | 13a | INH | = | 45 | % | ALA3802093 | % | Homo sapiens | |||
| 2. | ALA3800053 | 13a | INH | = | 55 | % | ALA3802092 | % | Homo sapiens | |||
| 3. | ALA3800053 | 13a | INH | = | 40 | % | ALA3802091 | % | Homo sapiens | |||
| 4. | ALA3800053 | 13a | CL | = | 1300 | ml/min.kg | ALA3802087 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 5. | ALA3800053 | 13a | Drug uptake | = | 0.5 | uM | ALA3802086 | uM | Rattus norvegicus | |||
| 6. | ALA3800053 | 13a | Cp | = | 28.3 | uM | ALA3802085 | uM | Rattus norvegicus | |||
| 7. | ALA3800053 | 13a | AUC | = | 14 | uM.hr | ALA3802084 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 8. | ALA3800053 | 13a | Cmax | = | 4.8 | uM | ALA3802083 | nM | Rattus norvegicus | |||
| 9. | ALA3800053 | 13a | F | = | 70 | % | ALA3802082 | % | Rattus norvegicus | |||
| 10. | ALA3800053 | 13a | t1/2 | = | 1.4 | hr | ALA3802081 | hr | Rattus norvegicus | |||
| 11. | ALA3800053 | 13a | CL | = | 47.5 | ml/min.kg | ALA3804655 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 12. | ALA3800053 | 13a | Ki | = | 776 | nM | ALA3804654 | 6.11 | nM | Homo sapiens | ||
| 13. | ALA3800053 | 13a | Ki | = | 3407 | nM | ALA3804653 | 5.47 | nM | Homo sapiens |
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