| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3800284 | 13e | INH | = | 45 | % | ALA3802093 | % | Homo sapiens | |||
| 2. | ALA3800284 | 13e | INH | = | 55 | % | ALA3802092 | % | Homo sapiens | |||
| 3. | ALA3800284 | 13e | INH | = | 40 | % | ALA3802091 | % | Homo sapiens | |||
| 4. | ALA3800284 | 13e | INH | = | 8 | uM | ALA3802090 | uM | Homo sapiens | |||
| 5. | ALA3800284 | 13e | CL | = | 3300 | ml/min.kg | ALA3802087 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 6. | ALA3800284 | 13e | Drug uptake | = | 0.07 | uM | ALA3802086 | uM | Rattus norvegicus | |||
| 7. | ALA3800284 | 13e | Cp | = | 5.65 | uM | ALA3802085 | uM | Rattus norvegicus | |||
| 8. | ALA3800284 | 13e | AUC | = | 19.7 | uM.hr | ALA3802084 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 9. | ALA3800284 | 13e | Cmax | = | 5.1 | uM | ALA3802083 | nM | Rattus norvegicus | |||
| 10. | ALA3800284 | 13e | F | = | 84 | % | ALA3802082 | % | Rattus norvegicus | |||
| 11. | ALA3800284 | 13e | t1/2 | = | 4.3 | hr | ALA3802081 | hr | Rattus norvegicus | |||
| 12. | ALA3800284 | 13e | CL | = | 22 | ml/min.kg | ALA3804655 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 13. | ALA3800284 | 13e | Ki | = | 64 | nM | ALA3804654 | 7.19 | nM | Homo sapiens | ||
| 14. | ALA3800284 | 13e | Ki | = | 174 | nM | ALA3804653 | 6.76 | nM | Homo sapiens |
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