# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3798468 | EPZ030456 | Ki | = | 4.7 | nM | ALA3803389 | 8.33 | nM | Homo sapiens | ||
2. | ALA3798468 | EPZ030456 | alphaKi | = | 1.1 | nM | ALA3803389 | nM | Homo sapiens | |||
3. | ALA3798468 | EPZ030456 | Ki | = | 1.3 | nM | ALA3803390 | 8.89 | nM | Homo sapiens | ||
4. | ALA3798468 | EPZ030456 | CLH | = | 34 | ml/min.kg | ALA3803392 | mL.min-1.kg-1 | ||||
5. | ALA3798468 | EPZ030456 | Papp | = | 0.34 | ucm/s | ALA3803393 | ucm/s | ||||
6. | ALA3798468 | EPZ030456 | Ratio | = | 104 | ALA3803394 | ||||||
7. | ALA3798468 | EPZ030456 | Fu | = | 0.32 | ALA3803395 | ||||||
8. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803122 | % | Homo sapiens | |||
9. | ALA3798468 | EPZ030456 | IC50 | = | 4 | nM | ALA3803119 | 8.40 | nM | Homo sapiens | ||
10. | ALA3798468 | EPZ030456 | IC50 | = | 48 | nM | ALA3803120 | 7.32 | nM | Homo sapiens | ||
11. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803121 | % | Homo sapiens | |||
12. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803123 | % | Homo sapiens | |||
13. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803124 | % | Homo sapiens | |||
14. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803125 | % | Homo sapiens | |||
15. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803126 | % | Homo sapiens | |||
16. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803127 | % | Homo sapiens | |||
17. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803128 | % | Homo sapiens | |||
18. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803129 | % | Homo sapiens | |||
19. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803130 | % | Homo sapiens | |||
20. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803382 | % | Homo sapiens |