# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3799220 | 14 | Ki | = | 13 | nM | ALA3801235 | 7.89 | nM | Homo sapiens | ||
2. | ALA3799220 | 14 | Ki | = | 74 | nM | ALA3801236 | 7.13 | nM | Homo sapiens | ||
3. | ALA3799220 | 14 | Ki | = | 38 | nM | ALA3801237 | 7.42 | nM | Homo sapiens | ||
4. | ALA3799220 | 14 | solubility | = | 126 | uM | ALA3801238 | nM | ||||
5. | ALA3799220 | 14 | Stability | = | 15 | % | ALA3801239 | % | Homo sapiens | |||
6. | ALA3799220 | 14 | Stability | = | 8 | % | ALA3801240 | % | ||||
7. | ALA3799220 | 14 | beta t1/2 | = | 0.62 | hr | ALA3801241 | hr | Mus musculus | |||
8. | ALA3799220 | 14 | CL | = | 3.92 | ml/min.kg | ALA3801242 | mL.min-1.kg-1 | Mus musculus | |||
9. | ALA3799220 | 14 | AUC | = | 13892 | ng.hr/ml | ALA3801243 | ng.hr.mL-1 | Mus musculus | |||
10. | ALA3799220 | 14 | F | = | 33 | % | ALA3801244 | % | Mus musculus | |||
11. | ALA3799220 | 14 | INH | = | 24 | % | ALA3801433 | % | Mus musculus | |||
12. | ALA3799220 | 14 | INH | 0 | ALA3801434 | Not Determined | % | Mus musculus | ||||
13. | ALA3799220 | 14 | INH | = | 21 | % | ALA3801435 | % | Mus musculus | |||
14. | ALA3799220 | 14 | INH | = | 31 | % | ALA3801436 | % | Mus musculus | |||
15. | ALA3799220 | 14 | INH | = | 58 | % | ALA3801437 | % | Mus musculus | |||
16. | ALA3799220 | 14 | Activity | 0 | ALA3801438 | Active | Mus musculus |