| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3797793 | 9a | pEC50 | = | 5.73 | ALA3804545 | 5.73 | nM | Rattus norvegicus | |||
| 2. | ALA3797793 | 9a | pEC50 | = | 6.14 | ALA3803186 | 6.14 | nM | Homo sapiens | |||
| 3. | ALA3797793 | 9a | FC | = | 5.4 | ALA3804562 | Homo sapiens | |||||
| 4. | ALA3797793 | 9a | EC50 | = | 180.6 | nM | ALA3804561 | 6.74 | nM | Homo sapiens | ||
| 5. | ALA3797793 | 9a | pEC50 | = | 6.74 | ALA3804560 | 6.74 | nM | Homo sapiens | |||
| 6. | ALA3797793 | 9a | Efficacy | = | 115.3 | % | ALA3804559 | % | Homo sapiens | |||
| 7. | ALA3797793 | 9a | Kp | = | 1.19 | ALA3804558 | ||||||
| 8. | ALA3797793 | 9a | Drug uptake | = | 83.6 | ng/g | ALA3804557 | ng/g | Rattus norvegicus | |||
| 9. | ALA3797793 | 9a | Cp | = | 80.2 | ng/ml | ALA3804556 | ng/ml | Rattus norvegicus | |||
| 10. | ALA3797793 | 9a | IC50 | > | 30 | uM | ALA3804555 | nM | Homo sapiens | |||
| 11. | ALA3797793 | 9a | IC50 | = | 2.9 | uM | ALA3804554 | 5.54 | nM | Homo sapiens | ||
| 12. | ALA3797793 | 9a | IC50 | = | 10.3 | uM | ALA3804553 | 4.99 | nM | Homo sapiens | ||
| 13. | ALA3797793 | 9a | IC50 | = | 2.9 | uM | ALA3804552 | 5.54 | nM | Homo sapiens | ||
| 14. | ALA3797793 | 9a | Fu | = | 0.017 | ALA3804551 | Rattus norvegicus | |||||
| 15. | ALA3797793 | 9a | Fu | = | 0.005 | ALA3804550 | Rattus norvegicus | |||||
| 16. | ALA3797793 | 9a | Fu | = | 0.027 | ALA3804549 | ||||||
| 17. | ALA3797793 | 9a | CLH | = | 62.2 | ml/min.kg | ALA3804548 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 18. | ALA3797793 | 9a | CLH | = | 9.85 | ml/min.kg | ALA3804547 | mL.min-1.kg-1 | Homo sapiens | |||
| 19. | ALA3797793 | 9a | %max | = | 124 | % | ALA3804546 | % | Rattus norvegicus | |||
| 20. | ALA3797793 | 9a | EC50 | = | 1.8 | uM | ALA3804545 | 5.75 | nM | Rattus norvegicus |
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