# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3814206 | 17 | t1/2 | = | 69 | min | ALA3855416 | hr | ||||
2. | ALA3814206 | 17 | t1/2 | = | 43 | min | ALA3855414 | hr | ||||
3. | ALA3814206 | 17 | IC50 | = | 608 | nM | ALA3855413 | 6.22 | nM | Homo sapiens | ||
4. | ALA3814206 | 17 | IC50 | > | 30000 | nM | ALA3855412 | nM | Homo sapiens | |||
5. | ALA3814206 | 17 | IC50 | = | 29450 | nM | ALA3855411 | 4.53 | nM | Homo sapiens | ||
6. | ALA3814206 | 17 | Efficacy | = | 56 | % | ALA3855410 | % | Homo sapiens | |||
7. | ALA3814206 | 17 | Efficacy | = | 60 | % | ALA3855409 | % | Homo sapiens | |||
8. | ALA3814206 | 17 | EC50 | = | 21 | nM | ALA3855408 | 7.68 | nM | Homo sapiens | ||
9. | ALA3814206 | 17 | EC50 | = | 244 | nM | ALA3855407 | 6.61 | nM | Homo sapiens | ||
10. | ALA3814206 | 17 | Ki | = | 3 | nM | ALA3855406 | 8.52 | nM | Homo sapiens | ||
11. | ALA3814206 | 17 | Ki | = | 81 | nM | ALA3855405 | 7.09 | nM | Homo sapiens | ||
12. | ALA3814206 | 17 | Efficacy | = | 56 | % | ALA3817101 | % | Homo sapiens | |||
13. | ALA3814206 | 17 | Efficacy | = | 60 | % | ALA3817100 | % | Homo sapiens | |||
14. | ALA3814206 | 17 | IC50 | = | 6600 | nM | ALA3817099 | 5.18 | nM | Homo sapiens | ||
15. | ALA3814206 | 17 | IC50 | 0 | ALA3817098 | Not Determined | Homo sapiens | |||||
16. | ALA3814206 | 17 | IC50 | = | 2200 | nM | ALA3817097 | 5.66 | nM | Homo sapiens | ||
17. | ALA3814206 | 17 | IC50 | = | 29430 | nM | ALA3817096 | 4.53 | nM | Homo sapiens | ||
18. | ALA3814206 | 17 | IC50 | > | 30000 | nM | ALA3817095 | nM | Homo sapiens | |||
19. | ALA3814206 | 17 | IC50 | = | 610 | nM | ALA3817094 | 6.21 | nM | Homo sapiens | ||
20. | ALA3814206 | 17 | t1/2 | = | 10 | min | ALA3817093 | hr | Macaca fascicularis |