# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3814815 | LY2955303 | inhibition | = | -0.19 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
2. | ALA3814815 | LY2955303 | Ki | > | 1700 | nM | ALA3817429 | nM | Homo sapiens | |||
3. | ALA3814815 | LY2955303 | Imax | > | 100 | % | ALA3817428 | % | Homo sapiens | |||
4. | ALA3814815 | LY2955303 | KB | = | 7.1 | nM | ALA3817427 | nM | Homo sapiens | |||
5. | ALA3814815 | LY2955303 | Ki | > | 2980 | nM | ALA3817430 | nM | Homo sapiens | |||
6. | ALA3814815 | LY2955303 | Ki | = | 1.1 | nM | ALA3817431 | 8.96 | nM | Homo sapiens | ||
7. | ALA3814815 | LY2955303 | Ratio Ki | > | 1560 | ALA3817432 | ||||||
8. | ALA3814815 | LY2955303 | solubility | > | 1 | mg/ml | ALA3817433 | ug.mL-1 | ||||
9. | ALA3814815 | LY2955303 | Ratio Ki | > | 2734 | ALA3817434 | ||||||
10. | ALA3814815 | LY2955303 | KB | > | 4440 | nM | ALA3817435 | nM | Homo sapiens | |||
11. | ALA3814815 | LY2955303 | KB | = | 1510 | nM | ALA3817436 | nM | Homo sapiens | |||
12. | ALA3814815 | LY2955303 | ED50 | = | 0.724 | mg kg-1 | ALA3817438 | mg.kg-1 | Rattus norvegicus | |||
13. | ALA3814815 | LY2955303 | AUC | = | 154 | ng.hr/ml | ALA3817439 | ng.hr.mL-1 | Rattus norvegicus | |||
14. | ALA3814815 | LY2955303 | AUC | = | 9100 | ng.hr/ml | ALA3817440 | ng.hr.mL-1 | Rattus norvegicus | |||
15. | ALA3814815 | LY2955303 | AUC | = | 36800 | ng.hr/ml | ALA3817441 | ng.hr.mL-1 | Rattus norvegicus | |||
16. | ALA3814815 | LY2955303 | Activity | 0 | ALA3817442 | Non-toxic | Rattus norvegicus | |||||
17. | ALA3814815 | LY2955303 | Activity | 0 | ALA3817533 | Toxic | Rattus norvegicus | |||||
18. | ALA3814815 | LY2955303 | F | = | 26 | % | ALA3817437 | % | Rattus norvegicus | |||
19. | ALA3814815 | LY2955303 | inhibition | = | -0.19 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
20. | ALA3814815 | LY2955303 | Inhibition | = | 14.03 | % | ALA4495582 | % | Severe acute respiratory syndrome coronavirus 2 |