# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3828396 | BRD4884 | Ratio | = | 7 | ALA3831142 | ||||||
2. | ALA3828396 | BRD4884 | AUC | = | 42 | /hr | ALA3830871 | /hr | Mus musculus | |||
3. | ALA3828396 | BRD4884 | Activity | = | 10 | % | ALA3830872 | % | Mus musculus | |||
4. | ALA3828396 | BRD4884 | INH | 0 | ALA3828960 | Active | % | Mus musculus | ||||
5. | ALA3828396 | BRD4884 | INH | 0 | ALA3828959 | Active | % | Mus musculus | ||||
6. | ALA3828396 | BRD4884 | AUC | = | 86 | /hr | ALA3828958 | /hr | Mus musculus | |||
7. | ALA3828396 | BRD4884 | Activity | = | 68 | % | ALA3828949 | % | Mus musculus | |||
8. | ALA3828396 | BRD4884 | K | = | 0.003 | /min | ALA3828948 | /min | Homo sapiens | |||
9. | ALA3828396 | BRD4884 | K | = | 0.001 | /min/microM | ALA3828941 | /min/microM | Homo sapiens | |||
10. | ALA3828396 | BRD4884 | K | = | 0.005 | /min | ALA3828947 | /min | Homo sapiens | |||
11. | ALA3828396 | BRD4884 | K | = | 0.014 | /min/microM | ALA3828946 | /min/microM | Homo sapiens | |||
12. | ALA3828396 | BRD4884 | K | = | 0.035 | /min | ALA3828945 | /min | Homo sapiens | |||
13. | ALA3828396 | BRD4884 | K | = | 0.41 | /min/microM | ALA3828944 | /min/microM | Homo sapiens | |||
14. | ALA3828396 | BRD4884 | Stability | = | 54 | % | ALA3828943 | % | ||||
15. | ALA3828396 | BRD4884 | Stability | = | 93 | % | ALA3828942 | % | Mus musculus | |||
16. | ALA3828396 | BRD4884 | t1/2 | = | 257 | min | ALA3830982 | hr | Homo sapiens | |||
17. | ALA3828396 | BRD4884 | IC50 | = | 1.09 | uM | ALA3830981 | 5.96 | nM | Homo sapiens | ||
18. | ALA3828396 | BRD4884 | Ki | = | 2.08 | uM | ALA3830981 | 5.68 | nM | Homo sapiens | ||
19. | ALA3828396 | BRD4884 | t1/2 | = | 143 | min | ALA3830980 | hr | Homo sapiens | |||
20. | ALA3828396 | BRD4884 | IC50 | = | 0.062 | uM | ALA3830979 | 7.21 | nM | Homo sapiens |