# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3827379 | 2; BMS-955176 | CC50 | = | 13 | uM | ALA5238914 | nM | Homo sapiens | |||
2. | ALA3827379 | 2; BMS-955176 | FC | = | 2 | ALA5238913 | ||||||
3. | ALA3827379 | 2; BMS-955176 | EC50 | = | 3 | nM | ALA5238911 | 8.52 | nM | Human immunodeficiency virus 1 | ||
4. | ALA3827379 | 2; BMS-955176 | EC50 | = | 700 | nM | ALA5238910 | 6.16 | nM | Human immunodeficiency virus 1 | ||
5. | ALA3827379 | 2; BMS-955176 | EC50 | = | 6 | nM | ALA5238909 | 8.22 | nM | Human immunodeficiency virus 1 | ||
6. | ALA3827379 | 2; BMS-955176 | EC50 | = | 6 | nM | ALA5238908 | 8.22 | nM | Human immunodeficiency virus 1 | ||
7. | ALA3827379 | 2; BMS-955176 | EC50 | = | 10 | nM | ALA5238907 | 8.00 | nM | Human immunodeficiency virus 1 | ||
8. | ALA3827379 | 2; BMS-955176 | EC50 | = | 5 | nM | ALA5238906 | 8.30 | nM | Human immunodeficiency virus 1 | ||
9. | ALA3827379 | 2; BMS-955176 | Ratio EC50 | = | 140 | ALA5119225 | ||||||
10. | ALA3827379 | 2; BMS-955176 | Ratio EC50 | > | 600 | ALA5119224 | ||||||
11. | ALA3827379 | 2; BMS-955176 | t1/2 | = | 43 | min | ALA5119223 | hr | ||||
12. | ALA3827379 | 2; BMS-955176 | Kd | = | 1.4 | nM | ALA5119222 | 8.85 | nM | |||
13. | ALA3827379 | 2; BMS-955176 | Activity | > | 1 | log10IU/ml | ALA5119216 | log10IU/ml | Human immunodeficiency virus 1 | |||
14. | ALA3827379 | 2; BMS-955176 | EC50 | > | 3 | uM | ALA5119197 | nM | Human immunodeficiency virus 1 | |||
15. | ALA3827379 | 2; BMS-955176 | Cmax | = | 0.1 | uM | ALA5119195 | nM | ||||
16. | ALA3827379 | 2; BMS-955176 | Cmax | = | 0.6 | uM | ALA5119194 | nM | ||||
17. | ALA3827379 | 2; BMS-955176 | Cmax | = | 1.2 | uM | ALA5119193 | nM | ||||
18. | ALA3827379 | 2; BMS-955176 | Cmax | = | 2.79 | uM | ALA5119192 | nM | ||||
19. | ALA3827379 | 2; BMS-955176 | AUCt | = | 1 | uM.hr | ALA5119191 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
20. | ALA3827379 | 2; BMS-955176 | AUCt | = | 29.3 | uM.hr | ALA5119190 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 |