| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3897426 | 50 | logKw | = | 0.52 | ALA3858003 | ||||||
| 2. | ALA3897426 | 50 | BPR | = | 0.5 | ALA3858001 | ||||||
| 3. | ALA3897426 | 50 | beta t1/2 | = | 1.02 | hr | ALA3858000 | hr | ||||
| 4. | ALA3897426 | 50 | Cmax | = | 515 | ng/ml | ALA3857969 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 5. | ALA3897426 | 50 | beta t1/2 | = | 1.07 | hr | ALA3857970 | hr | ||||
| 6. | ALA3897426 | 50 | Drug uptake | 0 | ALA3857999 | Active | ||||||
| 7. | ALA3897426 | 50 | Cmax | = | 1167 | ng/ml | ALA3857998 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 8. | ALA3897426 | 50 | Activity | 0 | ALA3857997 | Mus musculus | ||||||
| 9. | ALA3897426 | 50 | Activity | 0 | ALA3857995 | Mus musculus | ||||||
| 10. | ALA3897426 | 50 | Activity | 0 | ALA3857994 | Active | Mus musculus | |||||
| 11. | ALA3897426 | 50 | Activity | = | 130 | % | ALA3857993 | % | Mus musculus | |||
| 12. | ALA3897426 | 50 | Activity | = | 126 | % | ALA3857989 | % | Mus musculus | |||
| 13. | ALA3897426 | 50 | Activity | = | 124 | % | ALA3857988 | % | Mus musculus | |||
| 14. | ALA3897426 | 50 | CL | = | 16.1 | microL/min/mg | ALA3857984 | mL.min-1.g-1 | ||||
| 15. | ALA3897426 | 50 | t1/2 | = | 45 | min | ALA3857983 | hr | ||||
| 16. | ALA3897426 | 50 | Drug recovery | = | 27 | % | ALA3857976 | % | ||||
| 17. | ALA3897426 | 50 | Ki | = | 6.6 | nM | ALA3857975 | 8.18 | nM | |||
| 18. | ALA3897426 | 50 | Ki | = | 522 | nM | ALA3857974 | 6.28 | nM | Homo sapiens | ||
| 19. | ALA3897426 | 50 | Ki | = | 614 | nM | ALA3857973 | 6.21 | nM | Homo sapiens | ||
| 20. | ALA3897426 | 50 | Ki | = | 771 | nM | ALA3857972 | 6.11 | nM | Homo sapiens |
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