# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3897959 | 17d | INH | 0 | ALA3873644 | Dose-dependent effect | % | |||||
2. | ALA3897959 | 17d | Ratio IC50 | > | 1000 | ALA3873656 | ||||||
3. | ALA3897959 | 17d | INH | = | 0 | % | ALA3873655 | % | ||||
4. | ALA3897959 | 17d | INH | = | 0.5 | % | ALA3873654 | % | Homo sapiens | |||
5. | ALA3897959 | 17d | Ratio | = | 7 | ALA3873653 | ||||||
6. | ALA3897959 | 17d | Drug uptake | = | 13.12 | nM | ALA3873652 | nM | ||||
7. | ALA3897959 | 17d | Drug uptake | = | 2.32 | nM | ALA3873651 | nM | ||||
8. | ALA3897959 | 17d | Drug uptake | = | 2 | nM | ALA3873650 | nM | ||||
9. | ALA3897959 | 17d | Drug uptake | = | 0.62 | nM | ALA3873649 | nM | ||||
10. | ALA3897959 | 17d | Cp | = | 2867 | nM | ALA3873648 | nM | ||||
11. | ALA3897959 | 17d | Cp | = | 2162 | nM | ALA3873647 | nM | ||||
12. | ALA3897959 | 17d | Cp | = | 1054 | nM | ALA3873646 | nM | ||||
13. | ALA3897959 | 17d | Cp | = | 425 | nM | ALA3873645 | nM | ||||
14. | ALA3897959 | 17d | ED50 | = | 36.7 | mg kg-1 | ALA3873644 | mg.kg-1 | ||||
15. | ALA3897959 | 17d | INH | = | 73 | % | ALA3873643 | % | ||||
16. | ALA3897959 | 17d | INH | = | 65 | % | ALA3873642 | % | ||||
17. | ALA3897959 | 17d | INH | = | 43 | % | ALA3873641 | % | ||||
18. | ALA3897959 | 17d | INH | = | 13 | % | ALA3873640 | % | ||||
19. | ALA3897959 | 17d | INH | = | 65 | % | ALA3873638 | % | ||||
20. | ALA3897959 | 17d | INH | = | 80.2 | % | ALA3873637 | % | Homo sapiens |