# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3913540 | 30a | IC50 | = | 0.4 | nM | ALA3887609 | 9.40 | 344664 | nM | Homo sapiens | |
2. | ALA3913540 | 30a | IC50 | = | 0.1 | nM | ALA3887608 | 10.00 | 344595 | nM | Homo sapiens | |
3. | ALA3913540 | 30a | IC50 | = | 1.2 | uM | ALA3864816 | 5.92 | nM | Homo sapiens | ||
4. | ALA3913540 | 30a | F | = | 60 | % | ALA3864815 | % | ||||
5. | ALA3913540 | 30a | AUC | = | 3.2 | uM.hr | ALA3864814 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
6. | ALA3913540 | 30a | MRT | = | 4.3 | hr | ALA3864813 | hr | ||||
7. | ALA3913540 | 30a | Vdss | = | 6.7 | L/Kg | ALA3864812 | L.kg-1 | ||||
8. | ALA3913540 | 30a | CL | = | 1.6 | L/hr/kg | ALA3864811 | mL.min-1.kg-1 | ||||
9. | ALA3913540 | 30a | CLH | = | 33 | uL/min.mg | ALA3864810 | mL.min-1.g-1 | ||||
10. | ALA3913540 | 30a | CLH | = | 91 | uL/min.mg | ALA3864809 | mL.min-1.g-1 | ||||
11. | ALA3913540 | 30a | IC50 | = | 45 | nM | ALA3864807 | 7.35 | nM | Homo sapiens | ||
12. | ALA3913540 | 30a | IC50 | = | 0.43 | nM | ALA3864806 | 9.37 | nM | Homo sapiens | ||
13. | ALA3913540 | 30a | IC50 | = | 0.06 | nM | ALA3864805 | 10.22 | nM | Homo sapiens |