# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3928608 | 14 | TDI | = | 39 | % | ALA3858530 | % | Homo sapiens | |||
2. | ALA3928608 | 14 | F | = | 100 | % | ALA3858528 | % | ||||
3. | ALA3928608 | 14 | Cmax | = | 2050 | nM | ALA3858527 | nM | ||||
4. | ALA3928608 | 14 | Vdss | = | 2.3 | L/Kg | ALA3858526 | L.kg-1 | ||||
5. | ALA3928608 | 14 | t1/2 | = | 2.3 | hr | ALA3858525 | hr | ||||
6. | ALA3928608 | 14 | CL | = | 14 | ml/min.Kg | ALA3858524 | mL.min-1.kg-1 | ||||
7. | ALA3928608 | 14 | IC50 | = | 23 | nM | ALA3858523 | 7.64 | nM | Canis familiaris | ||
8. | ALA3928608 | 14 | IC50 | = | 11 | nM | ALA3858522 | 7.96 | nM | Canis familiaris | ||
9. | ALA3928608 | 14 | IC50 | = | 7.87 | uM | ALA3858521 | 5.10 | nM | |||
10. | ALA3928608 | 14 | Time | = | 24 | hr | ALA3858520 | hr | ||||
11. | ALA3928608 | 14 | F | = | 74 | % | ALA3858519 | % | ||||
12. | ALA3928608 | 14 | Vdss | = | 1.6 | L/Kg | ALA3858518 | L.kg-1 | ||||
13. | ALA3928608 | 14 | CL | = | 3.62 | ml/min.Kg | ALA3858517 | mL.min-1.kg-1 | ||||
14. | ALA3928608 | 14 | INH | = | 10 | % | ALA3858516 | % | Homo sapiens | |||
15. | ALA3928608 | 14 | INH | = | 0 | % | ALA3858515 | % | Homo sapiens | |||
16. | ALA3928608 | 14 | INH | = | 15 | % | ALA3858514 | % | Homo sapiens | |||
17. | ALA3928608 | 14 | Drug metabolism | = | 20 | % | ALA3858513 | % | ||||
18. | ALA3928608 | 14 | Drug metabolism | = | 13 | % | ALA3858512 | % | ||||
19. | ALA3928608 | 14 | Drug metabolism | = | 16 | % | ALA3858511 | % | ||||
20. | ALA3928608 | 14 | INH | 0 | ALA3858510 | % | Homo sapiens |