# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3932162 | 4; GSK5182 | IC50 | 0 | ALA4413880 | Not Determined | Homo sapiens | |||||
2. | ALA3932162 | 4; GSK5182 | Activity | 0 | ALA4413879 | Not Determined | ||||||
3. | ALA3932162 | 4; GSK5182 | Vdss | = | 16.8 | L/Kg | ALA4413831 | L.kg-1 | ||||
4. | ALA3932162 | 4; GSK5182 | CL | = | 44 | ml/min.kg | ALA4413828 | mL.min-1.kg-1 | ||||
5. | ALA3932162 | 4; GSK5182 | Cmax | = | 130 | nM | ALA4413827 | nM | ||||
6. | ALA3932162 | 4; GSK5182 | F | = | 8.4 | % | ALA4413826 | % | ||||
7. | ALA3932162 | 4; GSK5182 | AUC | = | 0.68 | uM.hr | ALA4413823 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
8. | ALA3932162 | 4; GSK5182 | IC50 | > | 30 | uM | ALA4413821 | nM | Homo sapiens | |||
9. | ALA3932162 | 4; GSK5182 | Peff | = | 0.23 | 10'-6 cm/s | ALA4413820 | 10'-6 cm/s | ||||
10. | ALA3932162 | 4; GSK5182 | Stability | = | 6.8 | % | ALA4413819 | % | ||||
11. | ALA3932162 | 4; GSK5182 | Stability | = | 26 | % | ALA4413818 | % | ||||
12. | ALA3932162 | 4; GSK5182 | Stability | = | 9.6 | % | ALA4413817 | % | ||||
13. | ALA3932162 | 4; GSK5182 | Stability | = | 42.8 | % | ALA4413816 | % | ||||
14. | ALA3932162 | 4; GSK5182 | INH | = | 17 | % | ALA4413815 | % | Homo sapiens | |||
15. | ALA3932162 | 4; GSK5182 | INH | = | 17.7 | % | ALA4413814 | % | Homo sapiens | |||
16. | ALA3932162 | 4; GSK5182 | INH | = | 21.8 | % | ALA4413813 | % | Homo sapiens | |||
17. | ALA3932162 | 4; GSK5182 | INH | = | 27.1 | % | ALA4413812 | % | Homo sapiens | |||
18. | ALA3932162 | 4; GSK5182 | INH | = | 16.4 | % | ALA4413811 | % | Homo sapiens | |||
19. | ALA3932162 | 4; GSK5182 | IC50 | = | 0.077 | uM | ALA4413810 | 7.11 | nM | Homo sapiens | ||
20. | ALA3932162 | 4; GSK5182 | IC50 | = | 2 | uM | ALA4413809 | 5.70 | nM | Homo sapiens |
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Standard Type
- IC50 12
- Activity 8
- Stability 8
- Inhibition 5
- AUC 1
- CL 1
- Cmax 1
- F 1
- Peff 1
- Vdss 1
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Organism Taxonomy L1
Organism Taxonomy L2
Organism Taxonomy L3
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- IC50 12
- result 9
- percent activity 7
- percent inhibition 5
- AUC 1
- CL 1
- Cmax 1
- F 1
- Vdss 1
- fold activation 1
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#RO5 Violations
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