| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3937708 | BDBM210802 | IC50 | = | 12 | nM | ALA3888090 | 7.92 | 372231 | nM | Homo sapiens | |
| 2. | ALA3937708 | BDBM210802 | INH | 0 | ALA5166443 | NA | % | Armoracia rusticana | ||||
| 3. | ALA3937708 | BDBM210802 | EC50 | = | 0.004 | uM | ALA5166394 | 8.38 | nM | Mus musculus | ||
| 4. | ALA3937708 | BDBM210802 | EC50 | = | 0.029 | uM | ALA5166393 | 7.54 | nM | Homo sapiens | ||
| 5. | ALA3937708 | BDBM210802 | K(p,uu,brain) | = | 0.01 | ALA5166392 | ||||||
| 6. | ALA3937708 | BDBM210802 | Fu | = | 0.02 | % | ALA5166391 | |||||
| 7. | ALA3937708 | BDBM210802 | Kp | = | 0.02 | ALA5166390 | ||||||
| 8. | ALA3937708 | BDBM210802 | F | = | 51 | % | ALA5166389 | % | ||||
| 9. | ALA3937708 | BDBM210802 | AUC/dose | = | 2407 | ng.hr/ml | ALA5166388 | ng.hr/ml | ||||
| 10. | ALA3937708 | BDBM210802 | t1/2 | = | 2.5 | hr | ALA5166387 | hr | ||||
| 11. | ALA3937708 | BDBM210802 | Vdss | = | 0.5 | L/Kg | ALA5166386 | L.kg-1 | ||||
| 12. | ALA3937708 | BDBM210802 | CL | = | 3.6 | ml/min.kg | ALA5166385 | mL.min-1.kg-1 | ||||
| 13. | ALA3937708 | BDBM210802 | Ratio | = | 0.8 | ALA5166384 | ||||||
| 14. | ALA3937708 | BDBM210802 | Papp | = | 53 | 10^-6 cm/s | ALA5166383 | 10^-6 cm/s | ||||
| 15. | ALA3937708 | BDBM210802 | IC50 | = | 0.017 | uM | ALA5166382 | 7.77 | nM | Homo sapiens | ||
| 16. | ALA3937708 | BDBM210802 | Fu | = | 0.1 | % | ALA5166381 |
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