# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3944154 | 10 | PB | = | 95.5 | % | ALA3868536 | % | Homo sapiens | |||
2. | ALA3944154 | 10 | PB | = | 86.6 | % | ALA3868535 | % | Homo sapiens | |||
3. | ALA3944154 | 10 | t1/2 | = | 5.6 | hr | ALA3868525 | hr | ||||
4. | ALA3944154 | 10 | CL | = | 8.4 | ml/min.kg | ALA3868524 | mL.min-1.kg-1 | ||||
5. | ALA3944154 | 10 | Efficacy | = | 47 | % | ALA3868521 | % | Homo sapiens | |||
6. | ALA3944154 | 10 | EC50 | = | 57 | nM | ALA3868520 | 7.24 | nM | Homo sapiens | ||
7. | ALA3944154 | 10 | Efficacy | = | 43 | % | ALA3868519 | % | Homo sapiens | |||
8. | ALA3944154 | 10 | EC50 | = | 8 | nM | ALA3868517 | 8.10 | nM | Homo sapiens | ||
9. | ALA3944154 | 10 | Ki | = | 10 | nM | ALA3868514 | 8.00 | nM | Homo sapiens | ||
10. | ALA3944154 | 10 | Ki | = | 53 | nM | ALA3868515 | 7.28 | nM | Homo sapiens | ||
11. | ALA3944154 | 10 | EC50 | = | 72 | nM | ALA3868513 | 7.14 | nM | Homo sapiens | ||
12. | ALA3944154 | 10 | Efficacy | = | 83 | % | ALA3868512 | % | Homo sapiens | |||
13. | ALA3944154 | 10 | Efficacy | = | 29 | % | ALA3868516 | % | Homo sapiens | |||
14. | ALA3944154 | 10 | EC50 | = | 76 | nM | ALA3868518 | 7.12 | nM | Homo sapiens |