| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  XL041 | BMS-852927 | Efficacy | = | 33 | % | ALA3868560 | % | Homo sapiens | |||
| 2. | XL041 | BMS-852927 | EC50 | = | 10 | nM | ALA3868559 | 8.00 | nM | Homo sapiens | ||
| 3. | XL041 | BMS-852927 | Activity | = | 8 | % | ALA3868557 | % | ||||
| 4. | XL041 | BMS-852927 | Activity | = | 20 | % | ALA3868556 | % | ||||
| 5. | XL041 | BMS-852927 | FC | = | 15 | ALA3868555 | Macaca fascicularis | |||||
| 6. | XL041 | BMS-852927 | FC | = | 4.7 | ALA3868554 | Macaca fascicularis | |||||
| 7. | XL041 | BMS-852927 | Cp | = | 22 | nM | ALA3868553 | nM | ||||
| 8. | XL041 | BMS-852927 | Cp | = | 7.5 | nM | ALA3868552 | nM | ||||
| 9. | XL041 | BMS-852927 | Activity | = | 10 | % | ALA3868550 | % | ||||
| 10. | XL041 | BMS-852927 | Cp | = | 57 | nM | ALA3868548 | nM | ||||
| 11. | XL041 | BMS-852927 | FC | = | 11 | ALA3868545 | Macaca fascicularis | |||||
| 12. | XL041 | BMS-852927 | Efficacy | = | 32 | % | ALA3868543 | % | ||||
| 13. | XL041 | BMS-852927 | EC50 | = | 5 | nM | ALA3868542 | 8.30 | nM | |||
| 14. | XL041 | BMS-852927 | betat1/2(app) | = | 10 | hr | ALA3868541 | hr | ||||
| 15. | XL041 | BMS-852927 | BPR | < | 0.05 | ALA3868540 | ||||||
| 16. | XL041 | BMS-852927 | Activity | = | 108 | % | ALA3868539 | % | Homo sapiens | |||
| 17. | XL041 | BMS-852927 | EC50 | = | 1 | uM | ALA3868528 | 6.00 | nM | Homo sapiens | ||
| 18. | XL041 | BMS-852927 | PB | = | 96.6 | % | ALA3868536 | % | Homo sapiens | |||
| 19. | XL041 | BMS-852927 | PB | = | 97.3 | % | ALA3868535 | % | Homo sapiens | |||
| 20. | XL041 | BMS-852927 | INH | 0 | ALA3868533 | % | Homo sapiens |
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