# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3953927 | 13 | betat1/2(app) | = | 10 | hr | ALA3868541 | hr | ||||
2. | ALA3953927 | 13 | Activity | = | 58 | % | ALA3868551 | % | ||||
3. | ALA3953927 | 13 | Activity | = | 2 | % | ALA3868550 | % | ||||
4. | ALA3953927 | 13 | Cp | = | 310 | nM | ALA3868549 | nM | ||||
5. | ALA3953927 | 13 | Cp | = | 85 | nM | ALA3868548 | nM | ||||
6. | ALA3953927 | 13 | FC | = | 10 | ALA3868547 | Macaca fascicularis | |||||
7. | ALA3953927 | 13 | FC | = | 4 | ALA3868545 | Macaca fascicularis | |||||
8. | ALA3953927 | 13 | Efficacy | = | 29 | % | ALA3868543 | % | ||||
9. | ALA3953927 | 13 | EC50 | = | 52 | nM | ALA3868542 | 7.28 | nM | |||
10. | ALA3953927 | 13 | Activity | = | 85 | % | ALA3868539 | % | Homo sapiens | |||
11. | ALA3953927 | 13 | EC50 | = | 3 | uM | ALA3868528 | 5.52 | nM | Homo sapiens | ||
12. | ALA3953927 | 13 | PB | = | 94.4 | % | ALA3868536 | % | Homo sapiens | |||
13. | ALA3953927 | 13 | PB | = | 87.6 | % | ALA3868535 | % | Homo sapiens | |||
14. | ALA3953927 | 13 | Efficacy | = | 34 | % | ALA3868521 | % | Homo sapiens | |||
15. | ALA3953927 | 13 | EC50 | = | 76 | nM | ALA3868520 | 7.12 | nM | Homo sapiens | ||
16. | ALA3953927 | 13 | Efficacy | = | 16 | % | ALA3868519 | % | Homo sapiens | |||
17. | ALA3953927 | 13 | EC50 | = | 8 | nM | ALA3868517 | 8.10 | nM | Homo sapiens | ||
18. | ALA3953927 | 13 | Efficacy | = | 12 | % | ALA3868516 | % | Homo sapiens | |||
19. | ALA3953927 | 13 | EC50 | = | 72 | nM | ALA3868518 | 7.14 | nM | Homo sapiens | ||
20. | ALA3953927 | 13 | Efficacy | = | 68 | % | ALA3868512 | % | Homo sapiens |