| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3955752 | 51 | INH | 0 | ALA3868371 | % | Rattus norvegicus | |||||
| 2. | ALA3955752 | 51 | Cmax | = | 24 | uM | ALA3868370 | nM | ||||
| 3. | ALA3955752 | 51 | Cmax | = | 5 | uM | ALA3868369 | nM | ||||
| 4. | ALA3955752 | 51 | Cmax | = | 0.73 | uM | ALA3868368 | nM | ||||
| 5. | ALA3955752 | 51 | AUC | = | 153 | uM.hr | ALA3868367 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 6. | ALA3955752 | 51 | AUC | = | 8.3 | uM.hr | ALA3868366 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 7. | ALA3955752 | 51 | AUC | = | 0.77 | uM.hr | ALA3868365 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 8. | ALA3955752 | 51 | Occ50 | = | 0.032 | uM | ALA3868364 | uM | Rattus norvegicus | |||
| 9. | ALA3955752 | 51 | K | = | 0.102 | /s | ALA3868363 | /s | Homo sapiens | |||
| 10. | ALA3955752 | 51 | K | = | 1.08 | 10'8/M/s | ALA3868362 | 10'8/M/s | Homo sapiens | |||
| 11. | ALA3955752 | 51 | Kd | = | 0.94 | nM | ALA3868361 | 9.03 | nM | Homo sapiens | ||
| 12. | ALA3955752 | 51 | PPB | = | 94 | % | ALA3868360 | % | ||||
| 13. | ALA3955752 | 51 | PPB | = | 92 | % | ALA3868359 | % | ||||
| 14. | ALA3955752 | 51 | Papp | = | 35 | 10'-6 cm/s | ALA3868358 | 10'-6 cm/s | ||||
| 15. | ALA3955752 | 51 | Ratio | = | 1 | ALA3868357 | ||||||
| 16. | ALA3955752 | 51 | F | = | 1 | % | ALA3868356 | % | ||||
| 17. | ALA3955752 | 51 | t1/2 | = | 0.8 | hr | ALA3868354 | hr | ||||
| 18. | ALA3955752 | 51 | CL | = | 33 | ml/min.kg | ALA3868353 | mL.min-1.kg-1 | ||||
| 19. | ALA3955752 | 51 | F | = | 37 | % | ALA3868352 | % | ||||
| 20. | ALA3955752 | 51 | t1/2 | = | 0.5 | hr | ALA3868351 | hr |
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