| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA339385 | Ap4A | INH | > | 50 | % | ALA5033287 | % | Homo sapiens | |||
| 2. | ALA339385 | Ap4A | Activity | = | 95 | % | ALA1817504 | % | ||||
| 3. | ALA339385 | Ap4A | Activity | = | 92.8 | % | ALA1817506 | % | ||||
| 4. | ALA339385 | Ap4A | Stability | = | 95 | % | ALA1817388 | % | ||||
| 5. | ALA339385 | Ap4A | Drug degradation | = | 17 | % | ALA1954472 | % | ||||
| 6. | ALA339385 | Ap4A | t1/2 | = | 4.4 | min | ALA3748146 | hr | Homo sapiens | |||
| 7. | ALA339385 | Ap4A | t1/2 | = | 2 | min | ALA3748147 | hr | Homo sapiens | |||
| 8. | ALA339385 | Ap4A | IC50 | < | 250 | uM | ALA3748153 | nM | Homo sapiens | |||
| 9. | ALA339385 | Ap4A | t1/2 | = | 2.99 | min | ALA3748143 | hr | Rattus norvegicus | |||
| 10. | ALA339385 | Ap4A | Activity | = | 198 | % | ALA3748119 | % | Homo sapiens | |||
| 11. | ALA339385 | Ap4A | t1/2 | = | 4.4 | min | ALA1067699 | hr | Rattus norvegicus | |||
| 12. | ALA339385 | Ap4A | t1/2 | = | 2 | min | ALA1068335 | hr | ||||
| 13. | ALA339385 | Ap4A | Ratio EC50 | = | 560 | ALA971528 | Homo sapiens | |||||
| 14. | ALA339385 | Ap4A | Ratio EC50 | = | 2 | ALA975343 | Homo sapiens | |||||
| 15. | ALA339385 | Ap4A | Efficacy | = | 12 | % | ALA971534 | % | Homo sapiens | |||
| 16. | ALA339385 | Ap4A | Efficacy | = | 117 | % | ALA974455 | % | Homo sapiens | |||
| 17. | ALA339385 | Ap4A | Efficacy | = | 149 | % | ALA974453 | % | Homo sapiens | |||
| 18. | ALA339385 | Ap4A | Efficacy | = | 68 | % | ALA971536 | % | Homo sapiens | |||
| 19. | ALA339385 | Ap4A | Efficacy | 0 | ALA975345 | Not Active | Homo sapiens | |||||
| 20. | ALA339385 | Ap4A | Efficacy | = | 68 | % | ALA974447 | % | Homo sapiens |
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