| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3973097 | 47 | Ki | = | 2143 | nM | ALA4731164 | 5.67 | nM | Homo sapiens | ||
| 2. | ALA3973097 | 47 | Ki | = | 5.2 | nM | ALA4731163 | 8.28 | nM | Homo sapiens | ||
| 3. | ALA3973097 | 47 | K | = | 0.21 | /s | ALA3868363 | /s | Homo sapiens | |||
| 4. | ALA3973097 | 47 | K | = | 4.43 | 10'7/M/s | ALA3868362 | 10'7/M/s | Homo sapiens | |||
| 5. | ALA3973097 | 47 | Kd | = | 4.74 | nM | ALA3868361 | 8.32 | nM | Homo sapiens | ||
| 6. | ALA3973097 | 47 | PPB | = | 84 | % | ALA3868360 | % | ||||
| 7. | ALA3973097 | 47 | PPB | = | 83 | % | ALA3868359 | % | ||||
| 8. | ALA3973097 | 47 | Papp | = | 33 | 10'-6 cm/s | ALA3868358 | 10'-6 cm/s | ||||
| 9. | ALA3973097 | 47 | Ratio | = | 1.1 | ALA3868357 | ||||||
| 10. | ALA3973097 | 47 | F | = | 16 | % | ALA3868355 | % | ||||
| 11. | ALA3973097 | 47 | t1/2 | = | 2 | hr | ALA3868354 | hr | ||||
| 12. | ALA3973097 | 47 | CL | = | 25 | ml/min.kg | ALA3868353 | mL.min-1.kg-1 | ||||
| 13. | ALA3973097 | 47 | F | = | 63 | % | ALA3868352 | % | ||||
| 14. | ALA3973097 | 47 | t1/2 | = | 1 | hr | ALA3868351 | hr | ||||
| 15. | ALA3973097 | 47 | CL | = | 12 | ml/min.kg | ALA3868350 | mL.min-1.kg-1 | ||||
| 16. | ALA3973097 | 47 | t1/2 | = | 3.2 | hr | ALA3868349 | hr | ||||
| 17. | ALA3973097 | 47 | CLH | = | 189 | ml/min.kg | ALA3868348 | mL.min-1.kg-1 | ||||
| 18. | ALA3973097 | 47 | CLH | < | 75 | ml/min.kg | ALA3868323 | mL.min-1.kg-1 | ||||
| 19. | ALA3973097 | 47 | CLH | = | 55 | ml/min.kg | ALA3868330 | mL.min-1.kg-1 | ||||
| 20. | ALA3973097 | 47 | IC50 | > | 10000 | nM | ALA3868324 | nM | Rattus norvegicus |
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