# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3979182 | BDBM238637 | t1/2 | = | 1.1 | hr | ALA4478478 | hr | ||||
2. | ALA3979182 | BDBM238637 | Vdss | = | 1.7 | L/Kg | ALA4478477 | L.kg-1 | ||||
3. | ALA3979182 | BDBM238637 | CL | = | 1.5 | L/hr/kg | ALA4478476 | mL.min-1.kg-1 | ||||
4. | ALA3979182 | BDBM238637 | CLH | = | 105 | microL/min/mg | ALA4478475 | mL.min-1.g-1 | ||||
5. | ALA3979182 | BDBM238637 | F | = | 54 | % | ALA4478472 | % | ||||
6. | ALA3979182 | BDBM238637 | t1/2 | = | 2.9 | hr | ALA4478471 | hr | ||||
7. | ALA3979182 | BDBM238637 | Vdss | = | 1.6 | L/Kg | ALA4478470 | L.kg-1 | ||||
8. | ALA3979182 | BDBM238637 | CL | = | 0.5 | L/hr/kg | ALA4478469 | mL.min-1.kg-1 | ||||
9. | ALA3979182 | BDBM238637 | CLH | = | 35 | microL/min/mg | ALA4478468 | mL.min-1.g-1 | ||||
10. | ALA3979182 | BDBM238637 | CLH | = | 52 | microL/min/mg | ALA4478467 | mL.min-1.g-1 | ||||
11. | ALA3979182 | BDBM238637 | IC50 | = | 29 | nM | ALA4478466 | 7.54 | nM | Homo sapiens | ||
12. | ALA3979182 | BDBM238637 | IC50 | = | 0.1 | nM | ALA4478465 | 10.00 | nM | Homo sapiens | ||
13. | ALA3979182 | BDBM238637 | IC50 | = | 0.1 | nM | ALA4478464 | 10.00 | nM | Homo sapiens | ||
14. | ALA3979182 | BDBM238637 | IC50 | = | 0.109 | nM | ALA3888800 | 9.96 | 416746 | nM | Homo sapiens | |
15. | ALA3979182 | BDBM238637 | IC50 | = | 0.116 | nM | ALA3888799 | 9.94 | 416426 | nM | Homo sapiens |